SCHEMBL4462480

SCHEMBL4462480

CCOC(=O)C1(COS(C)(=O)=O)CCC1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
POLB P06746 4/20 0.39
KMT2A Q03164 5/20 0.38
ALDH1A1 P00352 4/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
MEN1 O00255 4/20 0.35
KDM4E B2RXH2 2/20 0.34
LMNA P02545 1/20 0.33
GAA P10253 2/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL162359 0.93 ALDH1A1 (0.39) POLBKMT2AALDH1A1SMN1; SMN2MEN1
SCHEMBL716817 0.86 ALDH1A1 (0.36) POLBKMT2AALDH1A1SMN1; SMN2MEN1
SCHEMBL6950111 0.86 TSHR (0.39) POLBKMT2AALDH1A1MEN1LMNA
SCHEMBL12140577 0.86 ALDH1A1 (0.36) POLBKMT2AALDH1A1SMN1; SMN2MEN1
SCHEMBL20512092 0.85 POLB (0.38) POLBKMT2AALDH1A1SMN1; SMN2MEN1
SCHEMBL6777001 0.85 TSHR (0.36) POLBKMT2AALDH1A1SMN1; SMN2MEN1
SCHEMBL32670608 0.84 MAPT (0.41) POLBKMT2AALDH1A1SMN1; SMN2MEN1
SCHEMBL17540555 0.83 CYP4F2 (0.44) ALDH1A1KDM4ELMNA
SCHEMBL19209048 0.82 POLB (0.40) POLBKMT2AALDH1A1SMN1; SMN2KDM4E
SCHEMBL20512040 0.82 POLB (0.38) POLBKMT2AALDH1A1SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9242973-B2 Chromane compounds COMENTIS, INC. (US) 2016-01-26 US disclosed
US-9242973-B2 Chromane compounds COMENTIS, INC. (US) 2016-01-26 US disclosed
US-9242973-B2 Chromane compounds COMENTIS, INC. (US) 2016-01-26 US disclosed
US-20150225386-A1 CHROMANE COMPOUNDS COMENTIS, INC. 2015-08-13 US disclosed
US-20150225386-A1 CHROMANE COMPOUNDS COMENTIS, INC. 2015-08-13 US disclosed
US-8975415-B2 Chromane compounds COMENTIS, INC. (US) 2015-03-10 US disclosed
US-8975415-B2 Chromane compounds COMENTIS, INC. (US) 2015-03-10 US disclosed
US-8975415-B2 Chromane compounds COMENTIS, INC. (US) 2015-03-10 US disclosed
US-20140179695-A1 CHROMANE COMPOUNDS COMENTIS, INC. (US) 2014-06-26 US disclosed
US-20140179695-A1 CHROMANE COMPOUNDS COMENTIS, INC. (US) 2014-06-26 US disclosed
US-20140179695-A1 CHROMANE COMPOUNDS COMENTIS, INC. (US) 2014-06-26 US disclosed
WO-2013181202-A2 CHROMANE COMPOUNDS ASTELLAS PHARMA INC. (JP) 2013-12-05 WO disclosed
US-7576094-B2 Spiro derivatives as lipoxygenase inhibitors ELI LILLY AND COMPANY (US) 2009-08-18 US disclosed
EP-1836183-A2 SPIRO DERIVATIVES AS LIPOXYGENASE INHIBITORS Galileo Pharmaceuticals, Inc. (US) 2007-09-26 EP disclosed
WO-2006065686-A2 SPIRO DERIVATIVES AS LIPOXYGENASE INHIBITORS GALILEO PHARMACEUTICALS, INC. (US) 2006-06-22 WO disclosed
US-20060128790-A1 Spiro derivatives as lipoxygenase inhibitors GALILEO PHARMACEUTICALS, INC. 2006-06-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140179695-A1 CHROMANE COMPOUNDS BACE1, BACE2, APP POLB 1948/4885KMT2A 3884/4885ALDH1A1 4139/4885
US-20150225386-A1 CHROMANE COMPOUNDS BACE1, BACE2, APP POLB 2090/4885KMT2A 3037/4885ALDH1A1 3038/4885
US-20060128790-A1 Spiro derivatives as lipoxygenase inhibitors ALOX15B, ALOX5, ALOX15 POLB 2855/4885KMT2A 3967/4885ALDH1A1 169/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.