SCHEMBL4463073

SCHEMBL4463073

O=C(O)CCc1c[nH]c2ccc(F)cc12.OCCCc1c[nH]c2ccc(F)cc12

nearest known ligand 0.68

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MPO P05164 16/20 0.68
SLC6A4 P31645 6/20 0.68
TSHR P16473 1/20 0.63
HPGD P15428 1/20 0.60
CYP2C19 P33261 1/20 0.60
NOTUM Q6P988 2/20 0.55
MTNR1A P48039 1/20 0.55
MTNR1B P49286 1/20 0.55
HTR2A P28223 1/20 0.55
TRPM8 Q7Z2W7 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29902243 0.92 MPO (0.76) MPOSLC6A4TSHRHPGDCYP2C19
SCHEMBL3655654 0.92 MPO (0.76) MPOSLC6A4TSHRHPGDCYP2C19
SCHEMBL5203631 0.89 MPO (0.80) MPOSLC6A4TSHRNOTUMMTNR1A
SCHEMBL4352009 0.89 MPO (0.74) MPOSLC6A4HTR2ATRPM8
SCHEMBL5344966 0.88 MPO (0.80) MPOSLC6A4TSHRNOTUMMTNR1A
SCHEMBL5338627 0.87 MPO (0.78) MPOSLC6A4TSHRNOTUMMTNR1A
SCHEMBL5203031 0.85 MPO (0.73) MPOSLC6A4HTR2ATRPM8
SCHEMBL3702252 0.83 MPO (0.67) MPOSLC6A4NOTUMMTNR1AMTNR1B
SCHEMBL3695233 0.81 MPO (1.00) MPOSLC6A4TSHRNOTUMMTNR1A
SCHEMBL5637957 0.81 HTR2A (0.63) MPOSLC6A4TSHRHPGDCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009137733-A1 INDOLYLALKYL DERIVATIVES OF PYRIMIDINYLPIPERAZINE AND METABOLITES THEREOF FOR TREATMENT OF ANXIETY, DEPRESSION, AND SEXUAL DYSFUNCTION FABRE-KRAMER PHARMACEUTICALS, INC. (US) 2009-11-12 WO disclosed