SCHEMBL4463432

SCHEMBL4463432

O=C(O)N(c1ccccc1)c1ccc2cc[nH]c2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.50
ALDH1A1 P00352 2/20 0.50
ENPP2 Q13822 2/20 0.50
HPGD P15428 1/20 0.50
HSD17B10 Q99714 1/20 0.50
GHSR Q92847 2/20 0.44
TYR P14679 1/20 0.43
GLI1 P08151 1/20 0.42
GLI2 P10070 1/20 0.42
NLRP3 Q96P20 1/20 0.42
SLC6A2 P23975 2/20 0.41
SLC6A4 P31645 2/20 0.41
SLC6A3 Q01959 1/20 0.41
MAPK14 Q16539 1/20 0.40
MAPT P10636 1/20 0.40
AHR P35869 4/20 0.40
NPSR1 Q6W5P4 1/20 0.40
AGTR2 P50052 1/20 0.40
CYP2A6 P11509 1/20 0.40
TRPA1 O75762 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22418878 0.88 SLC6A2 (0.50) ENPP2GLI1GLI2SLC6A2SLC6A4
SCHEMBL14487695 0.78 ENPP2 (0.53) KDM4EALDH1A1ENPP2HPGDHSD17B10
SCHEMBL6166853 0.76 SLC6A2 (0.48) ENPP2GLI1GLI2SLC6A2SLC6A4
SCHEMBL19778 0.73 NPSR1 (0.70) ALDH1A1HPGDMAPTNPSR1
SCHEMBL15552410 0.73 RAB9A (0.55) KDM4EALDH1A1HPGD
SCHEMBL30026712 0.73 MAOA (0.64) KDM4EALDH1A1ENPP2HPGDHSD17B10
SCHEMBL27534535 0.72 ENPP2 (0.50) KDM4EALDH1A1ENPP2HPGDHSD17B10
SCHEMBL3425918 0.72 GLI1 (0.55) KDM4EALDH1A1ENPP2HPGDHSD17B10
Hydrochloric Acid SCHEMBL5094831 0.71 NPSR1 (0.67) ALDH1A1HPGDMAPTNPSR1
Bromide SCHEMBL31210017 0.71 NPSR1 (0.67) ALDH1A1HPGDMAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2035396-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY Synta Pharmaceuticals Corporation (US) 2009-03-18 EP disclosed
WO-2007139967-A2 TRIAZOLE COMPOUNDS THAT MODULATE HSP90 ACTIVITY SYNTA PHARMACEUTICALS CORP. (US) 2007-12-06 WO disclosed