SCHEMBL4465659

SCHEMBL4465659

COc1ccc(-n2c(N)c(N=O)c(=O)[nH]c2=S)cc1.COc1ccc(-n2c(N)cc(=O)[nH]c2=S)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.43
ATM Q13315 2/20 0.43
ALDH1A1 P00352 4/20 0.41
GAA P10253 1/20 0.41
MEN1 O00255 2/20 0.40
MAPT P10636 1/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KDM4E B2RXH2 1/20 0.39
PKM P14618 1/20 0.39
CA12 O43570 2/20 0.39
CA2 P00918 2/20 0.39
CA9 Q16790 2/20 0.39
CA1 P00915 1/20 0.39
LMNA P02545 1/20 0.38
PPARG P37231 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
NR2E3 Q9Y5X4 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
ESR2 Q92731 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4454976 0.91 KMT2A (0.50) KMT2AATMALDH1A1MEN1MAPT
SCHEMBL4495436 0.86 ATM (0.55) KMT2AATMALDH1A1GAAMEN1
SCHEMBL4460460 0.85 MAPT (0.51) KMT2AALDH1A1GAAMEN1MAPT
SCHEMBL4471377 0.79 GAA (0.52) KMT2AALDH1A1GAAMEN1MAPT
SCHEMBL4454534 0.78 GAA (0.48) KMT2AATMALDH1A1GAAMEN1
SCHEMBL4457582 0.76 KMT2A (0.55) KMT2AATMALDH1A1MEN1MAPT
SCHEMBL4492126 0.75 MAPT (0.47) KMT2AALDH1A1GAAMEN1MAPT
SCHEMBL7084232 0.73 ALDH1A1 (0.49) KMT2AALDH1A1GAAMEN1MAPT
SCHEMBL9381308 0.72 ATM (0.73) KMT2AATMALDH1A1GAAMEN1
SCHEMBL15331728 0.72 KMT2A (0.50) KMT2AATMALDH1A1MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010534-A1 THIOXANTHINE DERIVATIVES AND THEIR USE AS INHIBITORS OF MPO AstraZeneca AB (SE) 2009-01-07 EP disclosed
WO-2007120097-A1 THIOXANTHINE DERIVATIVES AND THEIR USE AS INHIBITORS OF MPO ASTRAZENECA AB (SE) 2007-10-25 WO disclosed