Trichostatin

Trichostatin

SCHEMBL446806

CC(/C=C/C(=O)NO)=C\C(C)C(=O)c1ccc(N(C)C)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 16/20 1.00
HDAC6 Q9UBN7 12/20 1.00
HDAC3 O15379 10/20 1.00
HDAC4 P56524 10/20 1.00
HDAC7 Q8WUI4 10/20 1.00
HDAC2 Q92769 10/20 1.00
HDAC10 Q969S8 10/20 1.00
HDAC8 Q9BY41 10/20 1.00
HDAC9 Q9UKV0 10/20 1.00
HDAC5 Q9UQL6 10/20 1.00
HDAC11 Q96DB2 9/20 1.00
CRHBP P24387 1/20 0.41
CRHR2 Q13324 1/20 0.41
TLR9 Q9NR96 1/20 0.41
TOP2A P11388 1/20 0.40
MAPT P10636 1/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trichostatin SCHEMBL446807 1.00 HDAC1 (1.00) HDAC1HDAC6HDAC3HDAC4HDAC7
Trichostatin SCHEMBL19886 1.00 HDAC1 (1.00) HDAC1HDAC6HDAC3HDAC4HDAC7
Trichostatin SCHEMBL675951 1.00 HDAC1 (1.00) HDAC1HDAC6HDAC3HDAC4HDAC7
Trichostatin SCHEMBL16380793 1.00 HDAC1 (1.00) HDAC1HDAC6HDAC3HDAC4HDAC7
Trichostatin SCHEMBL29450582 0.99 HDAC1 (0.97) HDAC1HDAC6HDAC3HDAC4HDAC7
SCHEMBL21965902 0.91 HDAC1 (0.83) HDAC1HDAC6HDAC3HDAC4HDAC7
SCHEMBL10324242 0.90 HDAC1 (0.81) HDAC1HDAC6HDAC3HDAC4HDAC7
SCHEMBL17119540 0.88 HDAC1 (0.79) HDAC1HDAC6HDAC3HDAC4HDAC7
SCHEMBL14392626 0.87 HDAC1 (0.77) HDAC1HDAC6HDAC3HDAC4HDAC7
SCHEMBL13301372 0.87 HDAC1 (0.77) HDAC1HDAC6HDAC3HDAC4HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 317 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260007676-A1 HDAC INHIBITORS FOR USE WITH NK CELL BASED THERAPIES VIRACTA THERAPEUTICS INC (US) 2026-01-08 US claimed
US-20240390375-A1 METHODS AND COMPOSITIONS FOR TREATING VIRAL OR VIRALLY-INDUCED CONDITIONS Viracta Subsidiary, Inc. (US) 2024-11-28 US claimed
WO-2024192348-A2 METHODS OF TREATING HPV IN HIV-INFECTED PATIENTS OHIO STATE INNOVATION FOUNDATION (US) 2024-09-19 WO claimed
US-20220249477-A1 METHODS AND COMPOSITIONS FOR TREATING VIRAL OR VIRALLY-INDUCED CONDITIONS VIRACTA THERAPEUTICS, INC. (US) 2022-08-11 US claimed
US-20200368280-A1 EPIGENETIC MODIFIERS FOR USE IN CELLULAR IMMUNOTHERAPY Viracta Subsidiary, Inc. 2020-11-26 US claimed
CN-110582564-A derivation of liver organoids from human pluripotent stem cells 新加坡科技研究局 2019-12-17 CN claimed
US-20190290646-A1 HDAC INHIBITORS FOR USE WITH NK CELL BASED THERAPIES INFINITY SA LLC, AS PURCHASER AGENT 2019-09-26 US claimed
EP-3484489-A1 HDAC INHIBITORS FOR USE WITH NK CELL BASED THERAPIES Viracta Therapeutics, Inc. (US) 2019-05-22 EP claimed
WO-2018013975-A1 HDAC INHIBITORS FOR USE WITH NK CELL BASED THERAPIES VIRACTA THERAPEUTICS, INC. (US) 2018-01-18 WO claimed
US-20150056192-A1 NOVEL COMPOSITIONS OF COMBINATIONS OF NON-COVALENT DNA BINDING AGENTS AND ANTI-CANCER AND/OR ANTI-INFLAMMATORY AGENTS AND THEIR USE IN DISEASE TREATMENT INDUS PHARMACEUTICALS, INC. 2015-02-26 US claimed
WO-2013151638-A1 NOVEL COMPOSITIONS OF COMBINATIONS OF NON-COVALENT DNA BINDING AGENTS AND ANTI-CANCER AND/OR ANTI-INFLAMMATORY AGENTS AND THEIR USE IN DISEASE TREATMENT INDUS PHARMACEUTICALS, INC. (US) 2013-10-10 WO claimed
US-20120141524-A1 ETHANOL EXTRACT OF ANTRODIA CAMPHORATA FOR INDUCING APOPTOSIS AND PREPARATION METHOD THEREOF KAOHSIUNG MEDICAL UNIVERSITY (TW) 2012-06-07 US claimed
US-20110245154-A1 Methods and Compositions for Treating Viral or Virally-Induced Conditions HEMAQUEST PHARMACEUTICALS, INC. (US) 2011-10-06 US claimed
WO-2011113013-A2 METHODS AND COMPOSITIONS FOR TREATING VIRAL OR VIRALLY-INDUCED CONDITIONS HEMAQUEST PHARMACEUTICALS, INC. (US) 2011-09-15 WO claimed
US-20100247543-A1 TREATMENT AND PREVENTION OF NEURODEGENERATIVE DISEASES ORYZON GENOMICS, S.A. (ES) 2010-09-30 US claimed
US-20100210869-A1 ETHANOL EXTRACT OF ANTRODIA CAMPHORATA FOR INDUCING APOPTOSIS AND PREPARATION METHOD THEREOF KAOHSIUNG MEDICAL UNIVERSITY (TW) 2010-08-19 US claimed
EP-2195029-A2 TREATMENT AND PREVENTION OF NEURODEGENERATIVE DISEASES Oryzon Genomics SA (ES) 2010-06-16 EP claimed
WO-2009027349-A2 TREATMENT AND PREVENTION OF NEURODEGENERATIVE DISEASES ORYZON GENOMICS SA (ES) 2009-03-05 WO claimed
WO-2008090534-A1 METHODS AND COMPOSITIONS FOR INHIBITION OF EXCESSIVE WEIGHT GAIN, REDUCTION OF INAPPROPRIATE EATING BEHAVIOURS AND INHIBITION OF BINGE EATING FOR THE TREATMENT OF OBESITY BERAND LIMITED (IE) 2008-07-31 WO claimed
WO-2007049262-A1 Methods and compositions for the promotion of neuronal growth and the treatment of asociality and affective disorders BERAND LIMITED (IE) 2007-05-03 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120141524-A1 ETHANOL EXTRACT OF ANTRODIA CAMPHORATA FOR INDUCING APOPTOSIS AND PREPARATION METHOD THEREOF BAX, API5, BCL2 HDAC1 1322/4885HDAC6 2916/4885HDAC3 1120/4885
US-20100210869-A1 ETHANOL EXTRACT OF ANTRODIA CAMPHORATA FOR INDUCING APOPTOSIS AND PREPARATION METHOD THEREOF BAX, API5, BCL2 HDAC1 1322/4885HDAC6 2916/4885HDAC3 1120/4885
US-20260007676-A1 HDAC INHIBITORS FOR USE WITH NK CELL BASED THERAPIES HDAC9, HDAC4, HDAC5 HDAC1 11/4885HDAC6 10/4885HDAC3 5/4885
US-20150056192-A1 NOVEL COMPOSITIONS OF COMBINATIONS OF NON-COVALENT DNA BINDING AGENTS AND ANTI-CANCER AND/OR ANTI-INFLAMMATORY AGENTS AND THEIR USE IN DISEASE TREATMENT TOP2A, HMGB1, TOP2B HDAC1 311/4885HDAC6 405/4885HDAC3 502/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.