SCHEMBL4468544

SCHEMBL4468544

CN(C)c1ccc(Cc2cnc(N)nc2N)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.62
PKM P14618 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11358841 0.84 DHFR (0.60) DHFR
SCHEMBL11286352 0.82 DHFR (0.68) DHFRPKM
SCHEMBL6557507 0.79 DHFR (0.58) DHFR
SCHEMBL28876908 0.79 DHFR (0.63) DHFR
SCHEMBL3937299 0.79 DHFR (0.68) DHFR
SCHEMBL8375784 0.79 DHFR (0.63) DHFR
SCHEMBL8380685 0.79 DHFR (0.63) DHFR
SCHEMBL380792 0.78 DHFR (0.67) DHFR
SCHEMBL11601563 0.78 DHFR (0.62) DHFRPKM
SCHEMBL8376680 0.78 DHFR (0.76) DHFRPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017838-A2 COMBINATIONS OF JAK-2 INHIBITORS AND OTHER AGENTS EXELIXIS, INC. (US) 2009-02-05 WO claimed
EP-0901473-A1 NOVEL PIPERAZINYLALKYLTHIOPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AND A PROCESS FOR THE PREPARATION OF THE NOVEL COMPOUNDS EGIS GYOGYSZERGYAR RT. (HU) 1999-03-17 EP disclosed
WO-1997016429-A1 NOVEL PIPERAZINYLALKYLTHIOPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AND A PROCESS FOR THE PREPARATION OF THE NOVEL COMPOUNDS EGIS Gyógyszergyár Rt. (HU) 1997-05-09 WO disclosed