SCHEMBL8375784

SCHEMBL8375784

Nc1ncc(Cc2ccc(Cl)cc2)c(N)n1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5669553 0.85 CSF1R (0.49) DHFR
SCHEMBL11286352 0.83 DHFR (0.68) DHFR
SCHEMBL3937299 0.83 DHFR (0.68) DHFR
SCHEMBL28876908 0.83 DHFR (0.63) DHFR
SCHEMBL8380685 0.83 DHFR (0.63) DHFR
SCHEMBL380792 0.82 DHFR (0.67) DHFR
SCHEMBL8380918 0.82 LMNA (0.66) DHFR
SCHEMBL8902607 0.82 DHFR (0.46) DHFR
SCHEMBL11271533 0.82 DHFR (0.62) DHFR
Water SCHEMBL28837029 0.81 DHFR (0.65) DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0901473-A1 NOVEL PIPERAZINYLALKYLTHIOPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AND A PROCESS FOR THE PREPARATION OF THE NOVEL COMPOUNDS EGIS GYOGYSZERGYAR RT. (HU) 1999-03-17 EP disclosed
WO-1997016429-A1 NOVEL PIPERAZINYLALKYLTHIOPYRIMIDINE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AND A PROCESS FOR THE PREPARATION OF THE NOVEL COMPOUNDS EGIS Gyógyszergyár Rt. (HU) 1997-05-09 WO disclosed
US-4315931-A MICROBIOCIDES, INFECTIOUS DISEASES BASF AKTIENGESELLSCHAFT (DE) 1982-02-16 US disclosed
EP-0000335-B1 ESTERS OF N-PYRIMIDINYL-CARBOXIMIDIC ACID, PROCESS FOR THEIR PREPARATION AND MEDICINES CONTAINING THEM. BASF Aktiengesellschaft (DE) 1981-10-07 EP disclosed
US-4279899-A MICROBIOCIDES BASF AKTIENGESELLSCHAFT (DE) 1981-07-21 US disclosed
US-4189581-A BACTERICIDES, POTENTIATORS OF SULFA DRUGS BASF AKTIENGESELLSCHAFT (DE) 1980-02-19 US disclosed
EP-0000334-A1 2,4-Diamino-5-benzyl-pyrimidines, process for their preparation and medicines containing them BASF Aktiengesellschaft (DE) 1979-01-24 EP disclosed