SCHEMBL4470461

SCHEMBL4470461

NC(=O)CCC(c1ccc(Cl)c(Cl)c1)N1CCNCC1

nearest known ligand 0.62

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 14/20 0.62
SLC6A4 P31645 14/20 0.62
TACR1 P25103 2/20 0.47
SLC6A3 Q01959 12/20 0.47
TNF P01375 1/20 0.44
OPRD1 P41143 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14775083 0.77 SLC6A4 (1.00) SLC6A2SLC6A4TACR1SLC6A3
SCHEMBL14775565 0.75 SLC6A4 (0.86) SLC6A2SLC6A4TACR1SLC6A3
SCHEMBL4483290 0.75 SLC6A2 (0.45) SLC6A2SLC6A4SLC6A3TNF
SCHEMBL13476435 0.72 SLC6A2 (0.62) SLC6A2SLC6A4TACR1SLC6A3OPRD1
SCHEMBL4470457 0.72 SIGMAR1 (0.49) SLC6A2SLC6A4TACR1SLC6A3
SCHEMBL13476431 0.72 SLC6A2 (0.59) SLC6A2SLC6A4TACR1SLC6A3OPRD1
SCHEMBL11079232 0.71 TNF (0.44) SLC6A2SLC6A4SLC6A3TNF
SCHEMBL4475063 0.69 TNF (0.45) SLC6A2SLC6A4SLC6A3TNF
SCHEMBL13476414 0.69 SLC6A2 (0.55) SLC6A2SLC6A4TACR1SLC6A3OPRD1
SCHEMBL13476463 0.69 SLC6A3 (0.60) SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7592344-B2 NK1 and NK2-antagonists and compositions and methods of using the same SOLVAY PHARMACEUTICALS GMBH (DE) 2009-09-22 US disclosed
EP-1954678-A1 NOVEL NK1 AND NK2 ANTAGONISTS Solvay Pharmaceuticals GmbH (DE) 2008-08-13 EP disclosed
US-20070149537-A1 NK1 and NK2-antagonists and compositions and methods of using the same SOLVAY PHARMACEUTICALS GMBH (DE) 2007-06-28 US disclosed
WO-2007063086-A1 NOVEL NK1 AND NK2 ANTAGONISTS SOLVAY PHARMACEUTICALS GMBH (DE) 2007-06-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070149537-A1 NK1 and NK2-antagonists and compositions and methods of using the same HRH2, PROKR2, BDKRB2 SLC6A2 1388/4885SLC6A4 2566/4885TACR1 9/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.