SCHEMBL4472284

SCHEMBL4472284

N#Cc1cccc(S(=O)(=O)NC(=O)c2ccccc2N)c1

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KAT6A Q92794 4/20 0.58
FLT1 P17948 5/20 0.48
FLT4 P35916 5/20 0.48
KDR P35968 5/20 0.48
KDM4E B2RXH2 2/20 0.46
PGR P06401 1/20 0.45
HPGD P15428 1/20 0.45
HTT P42858 1/20 0.43
ACLY P53396 2/20 0.43
PTGES2 Q9H7Z7 1/20 0.43
RXFP1 Q9HBX9 1/20 0.42
CCKBR P32239 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4196234 0.80 KDM4E (0.68) FLT1FLT4KDRKDM4EHPGD
SCHEMBL4477897 0.80 FLT1 (0.67) KAT6AFLT1FLT4KDRKDM4E
SCHEMBL6850238 0.77 KAT6A (0.51) KAT6AKDM4EPGRACLYPTGES2
SCHEMBL17127741 0.76 KAT6A (0.53) KAT6APGRACLYRXFP1CCKBR
SCHEMBL5666232 0.76 HTT (0.72) HTTRXFP1
SCHEMBL5958934 0.76 FLT1 (0.65) KAT6AFLT1FLT4KDRRXFP1
SCHEMBL4476657 0.75 HPGD (0.55) KAT6AFLT1FLT4KDRKDM4E
SCHEMBL4472286 0.74 CYP2C9 (0.58) KAT6APGRHTTACLY
SCHEMBL19006934 0.73 KAT6A (0.50) KAT6APGRACLYPTGES2RXFP1
SCHEMBL420253 0.73 PGR (0.54) KAT6APGRACLYPTGES2RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009067607-A2 COMBINATIONS OF PDE4 INHIBITORS AND ANTIPSYCHOTICS FOR THE TREATMENT OF PSYCHOTIC DISORDERS MEMORY PHARMACEUTICALS CORPORATION (US) 2009-05-28 WO disclosed