SCHEMBL4473387

SCHEMBL4473387

Cc1nc(N)nc(N)c1-c1cc(C2CC2)n[nH]1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DHFR P00374 3/20 0.35
HRH4 Q9H3N8 3/20 0.35
PDE8B O95263 1/20 0.34
HRH3 Q9Y5N1 1/20 0.33
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32
HPGD P15428 1/20 0.32
NUDT1 P36639 1/20 0.32
HSD17B10 Q99714 1/20 0.32
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
PIK3CA P42336 3/20 0.31
DRD2 P14416 1/20 0.31
DRD4 P21917 1/20 0.31
DRD3 P35462 1/20 0.31
MTOR P42345 1/20 0.31
HEXA P06865 1/20 0.31
HEXB P07686 1/20 0.31
ILK Q13418 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4455888 0.78 HCAR2 (0.43) DHFRCYP1A2DRD4
SCHEMBL1792501 0.74 IGF1R (0.52)
SCHEMBL4074269 0.73 NTRK1 (0.49)
SCHEMBL4469628 0.72 ADORA2A (0.41) DHFRPDE8BPIK3CA
SCHEMBL4470547 0.71 CDC7 (0.33) HRH4PDE8BHRH3
SCHEMBL30782745 0.68 HRH4 (0.40) DHFRHRH4HRH3PIK3CA
SCHEMBL31663246 0.67 KMT2A (0.40) HRH4ALDH1A1CYP1A2HSD17B10
SCHEMBL25338891 0.66 ALDH1A1 (0.42) ALDH1A1
SCHEMBL14722727 0.66 HCAR2 (0.42) ALDH1A1CYP1A2DRD4
SCHEMBL170833 0.65

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017838-A2 COMBINATIONS OF JAK-2 INHIBITORS AND OTHER AGENTS EXELIXIS, INC. (US) 2009-02-05 WO claimed