SCHEMBL4469628

SCHEMBL4469628

Nc1ncc(-c2cc(C3CC3)n[nH]2)c(N)n1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.41
ADORA1 P30542 1/20 0.41
DHFR P00374 9/20 0.40
PIK3CA P42336 1/20 0.35
PDE8B O95263 1/20 0.34
RET P07949 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30782745 0.94 HRH4 (0.40) ADORA2AADORA1DHFRPIK3CA
SCHEMBL4464801 0.78 DHFR (0.42) ADORA1DHFR
SCHEMBL4457723 0.77 HCAR2 (0.43) ADORA2AADORA1DHFRPIK3CA
SCHEMBL4077928 0.73 NTRK1 (0.49)
SCHEMBL4466340 0.73 IGF1R (0.50) ADORA2AADORA1
SCHEMBL3941063 0.73 NTRK1 (0.52)
SCHEMBL4473387 0.72 DHFR (0.35) DHFRPIK3CAPDE8B
SCHEMBL23217059 0.72 NTRK1 (0.52)
SCHEMBL28664537 0.71 MKNK1 (0.40) ADORA2AADORA1DHFRPIK3CA
SCHEMBL4470547 0.70 CDC7 (0.33) ADORA2AADORA1PDE8B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009017838-A2 COMBINATIONS OF JAK-2 INHIBITORS AND OTHER AGENTS EXELIXIS, INC. (US) 2009-02-05 WO claimed