SCHEMBL4479458

SCHEMBL4479458

CC(=O)Oc1cccc2cc(S(=O)(=O)NCc3cccc4ccccc34)ccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.45
POLB P06746 2/20 0.44
HSD17B10 Q99714 2/20 0.44
MEN1 O00255 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2C9 P11712 1/20 0.44
KMT2A Q03164 1/20 0.44
ALDH1A1 P00352 2/20 0.44
TP53 P04637 2/20 0.44
CYP19A1 P11511 1/20 0.43
MAPK1 P28482 2/20 0.42
GAA P10253 2/20 0.42
PGR P06401 1/20 0.42
PTGS1 P23219 1/20 0.42
THRB P10828 1/20 0.42
HTR6 P50406 2/20 0.41
NQO2 P16083 1/20 0.41
MTNR1A P48039 1/20 0.41
MAPT P10636 1/20 0.41
HTT P42858 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4482883 0.87 CYP19A1 (0.53) POLBCYP1A2KMT2AALDH1A1CYP19A1
SCHEMBL4485797 0.86 POLB (0.48) POLBHSD17B10MEN1CYP1A2CYP2C9
SCHEMBL4478333 0.83 ALDH1A1 (0.50) MEN1CYP1A2CYP2C9KMT2AALDH1A1
SCHEMBL4482164 0.82 ATM (0.54) POLBALDH1A1GAAHTTL3MBTL1
SCHEMBL4483653 0.81 CYP19A1 (0.53) POLBCYP19A1MAPK1
SCHEMBL4471125 0.80 LMNA (0.51) POLBHSD17B10MEN1KMT2AALDH1A1
SCHEMBL4471119 0.80 AKR1C3 (0.53) POLBMEN1KMT2AALDH1A1GAA
SCHEMBL4478162 0.80 CA2 (0.56) CA2POLBHSD17B10MEN1CYP1A2
SCHEMBL4477096 0.80 POLB (0.39) POLBALDH1A1CYP19A1GAAHTR6
SCHEMBL4472720 0.80 HDAC3 (0.51) POLBALDH1A1CYP19A1GAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7598418-B2 Naphthalene-1-(sulfonamide or carboxamide) derivatives; e.g. N-Benzyl-5-{[(4-methylphenyl)sulfonyl]oxy}naphthalene-1-sulfonamide; protein kinase inhibitors sensitize cancer cells to radiotherapy or anticancer agents; side effect reduction INSTITUTE OF MEDICINAL MOLECULAR DESIGN, INC. (JP) 2009-10-06 US claimed
US-20050215645-A1 Amide derivatives INSTITUTE OF MEDICINAL MOLECULAR DESIGN. INC. (JP) 2005-09-29 US claimed
US-7598418-B2 Naphthalene-1-(sulfonamide or carboxamide) derivatives; e.g. N-Benzyl-5-{[(4-methylphenyl)sulfonyl]oxy}naphthalene-1-sulfonamide; protein kinase inhibitors sensitize cancer cells to radiotherapy or anticancer agents; side effect reduction INSTITUTE OF MEDICINAL MOLECULAR DESIGN, INC. (JP) 2009-10-06 US disclosed
US-20050215645-A1 Amide derivatives INSTITUTE OF MEDICINAL MOLECULAR DESIGN. INC. (JP) 2005-09-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050215645-A1 Amide derivatives OGG1, HDAC1, BCL2A1 CA2 926/4885POLB 296/4885HSD17B10 2044/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.