SCHEMBL4483103

SCHEMBL4483103

CCNC(=O)N1CCC(NC(=O)OCc2ccccc2)C(C(c2ccc(F)cc2)c2ccc(F)cc2)C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 3/20 0.46
DPP4 P27487 6/20 0.45
DPP7 Q9UHL4 6/20 0.45
KCNH2 Q12809 4/20 0.45
TSHR P16473 2/20 0.44
FAAH O00519 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
ALOX12 P18054 1/20 0.44
MAPK1 P28482 1/20 0.44
MTOR P42345 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
MEN1 O00255 1/20 0.43
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43
KMT2A Q03164 1/20 0.43
ALDH1A1 P00352 1/20 0.41
CPB1 P15086 2/20 0.41
CTSL P07711 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4483695 0.85 P2RX7 (0.47) CTSKDPP4DPP7KCNH2MAPK1
SCHEMBL4483683 0.85 P2RX7 (0.47) CTSKDPP4DPP7KCNH2MAPK1
SCHEMBL4483688 0.85 P2RX7 (0.47) CTSKDPP4DPP7KCNH2MAPK1
Trifluoroacetic Acid SCHEMBL4484957 0.73 DPP4 (0.44) DPP4DPP7KCNH2TSHRFAAH
Trifluoroacetic Acid SCHEMBL4484950 0.73 DPP4 (0.44) DPP4DPP7KCNH2TSHRFAAH
Hydrochloric Acid SCHEMBL4480328 0.71 KMT2A (0.59) DPP4DPP7TSHRFAAHCYP3A4
SCHEMBL29268591 0.71 CTSK (0.60) CTSKDPP4DPP7KCNH2TSHR
SCHEMBL21522663 0.71 CTSK (0.60) CTSKDPP4DPP7KCNH2TSHR
SCHEMBL29268593 0.71 CTSK (0.60) CTSKDPP4DPP7KCNH2TSHR
SCHEMBL5943236 0.71 PREP (0.44) CTSKTSHRCYP3A4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7622487-B2 Piperidine derivative, process for producing the same, and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-11-24 US disclosed