SCHEMBL4495798

SCHEMBL4495798

COC(=O)c1cccc(-c2[nH]c(C=O)c(C(=O)O)c2C(C)C)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 5/20 0.46
KDM5B Q9UGL1 1/20 0.45
ALDH1A1 P00352 3/20 0.44
RAB9A P51151 1/20 0.44
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39
GABRA5 P31644 1/20 0.39
GABRA3 P34903 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA9 Q16790 1/20 0.39
SLC7A5 Q01650 1/20 0.39
CDK8 P49336 1/20 0.38
NEK1 Q96PY6 1/20 0.38
AXL P30530 1/20 0.38
HCRTR1 O43613 1/20 0.38
HCRTR2 O43614 1/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4495480 0.86 ALDH1A1 (0.42) ERN1KDM5BALDH1A1RAB9ACA12
SCHEMBL4491011 0.82 SMN1; SMN2 (0.44) ALDH1A1RAB9AMAPTKMT2ASMN1; SMN2
SCHEMBL4495792 0.77 ERN1 (0.47) ERN1ALDH1A1RAB9ACA12CA1
SCHEMBL4492959 0.72 CA12 (0.41) ERN1ALDH1A1RAB9ACA12CA1
SCHEMBL4485738 0.72 MTNR1A (0.41) ALDH1A1POLBKMT2A
SCHEMBL4504198 0.71 LDHA (0.38) KDM5BALDH1A1POLBMAPTBLM
SCHEMBL20074249 0.71 KDM5B (0.54) ERN1KDM5BALDH1A1GABRG2GABRB3
SCHEMBL31676974 0.71 KDM5B (0.54) ERN1KDM5BALDH1A1GABRG2GABRB3
SCHEMBL4491747 0.70 MEN1 (0.40) ALDH1A1RAB9APOLBMAPTKMT2A
SCHEMBL4496742 0.70 CCR1 (0.36) ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504429-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2009-03-17 US claimed