SCHEMBL4495480

SCHEMBL4495480

COC(=O)c1ccc(-c2[nH]c(C=O)c(C(=O)O)c2C(C)C)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
RAB9A P51151 2/20 0.41
KDM5B Q9UGL1 1/20 0.41
ERN1 O75460 3/20 0.40
RAF1 P04049 1/20 0.38
IDO1 P14902 1/20 0.37
KDM4E B2RXH2 2/20 0.36
TSHR P16473 1/20 0.36
TNKS O95271 1/20 0.36
TLR9 Q9NR96 1/20 0.36
TLR8 Q9NR97 1/20 0.36
TLR7 Q9NYK1 1/20 0.36
PTPN1 P18031 1/20 0.36
STAT3 P40763 1/20 0.36
NPC1 O15118 1/20 0.36
LMNA P02545 1/20 0.36
PKM P14618 1/20 0.36
HPGD P15428 1/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4495798 0.86 ERN1 (0.46) ALDH1A1RAB9AKDM5BERN1SMN1; SMN2
SCHEMBL4491747 0.78 MEN1 (0.40) ALDH1A1RAB9APKMSMN1; SMN2TDP1
SCHEMBL4488479 0.75 ALDH1A1 (0.44) ALDH1A1RAB9AERN1RAF1KDM4E
SCHEMBL4492959 0.73 CA12 (0.41) ALDH1A1RAB9AERN1KDM4ELMNA
SCHEMBL4497716 0.71 BTK (0.41)
SCHEMBL4490045 0.71 PPARG (0.42) ALDH1A1RAB9AKDM4EHPGDSMN1; SMN2
SCHEMBL4488655 0.70 KDM4E (0.36) ALDH1A1KDM5BERN1KDM4ELMNA
SCHEMBL4504198 0.70 LDHA (0.38) ALDH1A1KDM5BKDM4ETLR9TLR8
SCHEMBL4494581 0.69 ESR1 (0.38) ALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL4492341 0.69 LDHA (0.36) ALDH1A1KDM4ENPC1LMNAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504429-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2009-03-17 US claimed