SCHEMBL449631

SCHEMBL449631

[c]1ccc2cc[c]nc2c1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL196535 0.84
SCHEMBL2910 0.73 CYP1A2 (0.44)
SCHEMBL4315969 0.71
SCHEMBL9322559 0.70 ACHE (0.42)
SCHEMBL1450761 0.70 CYP1A2 (0.52)
SCHEMBL6360076 0.69
SCHEMBL198099 0.68
SCHEMBL452557 0.68
SCHEMBL16316 0.68 MAP4K4 (0.34)
SCHEMBL4843118 0.68 BACE1 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230210840-A1 BACTERIAL NITRIC OXIDE SYNTHASE INHIBITORS NORTHWESTERN UNIVERSITY 2023-07-06 US disclosed
CN-114805831-A Metal organic material and preparation method 耶达研究及发展有限公司 2022-07-29 CN disclosed
CN-113166098-A Triazine compound, material for organic electroluminescent element, and organic electroluminescent element 东曹株式会社 2021-07-23 CN disclosed
US-9707540-B2 Metal-organic materials and method for preparation YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2017-07-18 US disclosed
US-9611218-B2 Metal-organic materials and method for preparation YEDA RESEARCH AND DEVELOPMENT CO., LTD. (IL) 2017-04-04 US disclosed
US-20160271582-A1 METAL-ORGANIC MATERIALS AND METHOD FOR PREPARATION YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2016-09-22 US disclosed
CN-105873987-A Metal organic material and preparation method 耶达研究及发展有限公司 2016-08-17 CN disclosed
US-20160152568-A1 METAL-ORGANIC MATERIALS AND METHOD FOR PREPARATION YEDA RESEARCH AND DEVELOPMENT CO. LTD. (IL) 2016-06-02 US disclosed
EP-3022250-A1 METAL-ORGANIC MATERIALS AND METHOD FOR PREPARATION YEDA RESEARCH AND DEVELOPMENT CO. LTD., AT THE WEI (IL) 2016-05-25 EP disclosed
US-20150216861-A1 CYCLOPROPYL AMIDE DERIVATIVES ASTRAZENECA AB (SE) 2015-08-06 US disclosed
EP-2195293-A2 CYCLOPTOPYL AMIDE DERIVATIVES AstraZeneca AB (SE) 2010-06-16 EP disclosed
WO-2010062245-A1 SPIROCYCLOBUTYL PIPERIDINE DERIVATIVES ASTRAZENECA AB (SE) 2010-06-03 WO disclosed
US-20100130477-A1 Spirocyclobutyl Piperidine Derivatives ASTRAZENECA AB (SE) 2010-05-27 US disclosed
US-20090076020-A1 Cyclopropyl Amide Derivatives 978 ASTRAZENECA AB (SE) 2009-03-19 US disclosed
WO-2009024823-A2 OXADIAZOLE DERIVATIVES AS DGAT INHIBITORS ASTRAZENECA AB (SE) 2009-02-26 WO disclosed
US-20050085447-A1 Pyrido[3,4-d]pyrimidine derivatives as matrix metalloproteinase-13 inhibitors WARNER-LAMBERT COMPANY LLC 2005-04-21 US disclosed
WO-2005016926-A1 PYRIDO [3,4-D] PYRIMIDINE DERIVATIVES AS MATRIX METALLOPROTEINASE-13 INHIBITORS WARNER-LAMBERT COMPANY LLC (US) 2005-02-24 WO disclosed
US-6166210-A Perylene imide monocarboxylic acids CIBA SPECIALTY CHEMICALS CORPORATION (US) 2000-12-26 US disclosed
EP-1053228-A1 PERYLENE IMIDE MONOCARBOXYLIC ACIDS AS COLORANTS Ciba SC Holding AG (CH) 2000-11-22 EP disclosed
WO-1999031069-A1 PERYLENE IMIDE MONOCARBOXYLIC ACIDS AS COLORANTS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 1999-06-24 WO disclosed