SCHEMBL4496901

SCHEMBL4496901

CC(C)N1CCN(c2ccc(N)c(F)c2)C(=O)C1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 5/20 0.40
KCNH2 Q12809 5/20 0.40
HRH3 Q9Y5N1 4/20 0.37
SLC6A2 P23975 4/20 0.35
SLC6A4 P31645 2/20 0.35
BPTF Q12830 1/20 0.35
DRD2 P14416 4/20 0.34
CACNA2D1 P54289 3/20 0.33
PARP1 P09874 1/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4496899 0.83 HRH3 (0.44) DRD3KCNH2HRH3PARP1
SCHEMBL3973870 0.79 HRH3 (0.41) HRH3PARP1ALDH1A1KDM4EMAPT
SCHEMBL22171249 0.78 MAPT (0.51) HRH3ALDH1A1KDM4EMAPTPKM
SCHEMBL3974009 0.77 DDB1 (0.46) DRD3KCNH2SLC6A2DRD2CACNA2D1
Hydrochloric Acid SCHEMBL22165259 0.77 MAPT (0.50) HRH3ALDH1A1KDM4EMAPTPKM
SCHEMBL23176630 0.76 LMNA (0.44) DRD3KCNH2HRH3DRD2ALDH1A1
SCHEMBL13256438 0.74 NPC1 (0.50) DRD3KCNH2HRH3DRD2PARP1
SCHEMBL4079481 0.73 SIRT6 (0.44) KCNH2ALDH1A1KDM4EMAPTPKM
SCHEMBL17055336 0.73 HRH3 (0.39) DRD3KCNH2HRH3PARP1ALDH1A1
SCHEMBL3551615 0.73 ALDH1A1 (0.50) ALDH1A1KDM4EPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7601752-B2 Pyrrolidine derivatives HOFFMANN-LA ROCHE INC. (US) 2009-10-13 US disclosed
US-20070112001-A1 Pyrrolidine derivatives F. HOFFMANN-LA ROCHE AG, A SWISS COMPANY (CH) 2007-05-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070112001-A1 Pyrrolidine derivatives F12, F2, F11 DRD3 985/4885KCNH2 1383/4885HRH3 497/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.