SCHEMBL4497666

SCHEMBL4497666

CC(C)C(=O)Nc1n[nH]c2cc(-c3cccc(F)c3)ccc12

nearest known ligand 0.69

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 8/20 0.69
GSK3A P49840 3/20 0.69
AAK1 Q2M2I8 7/20 0.63
CYP1A2 P05177 1/20 0.57
HDAC6 Q9UBN7 4/20 0.53
GAK O14976 1/20 0.52
STK16 O75716 1/20 0.52
BMP2K Q9NSY1 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4491027 0.89 GSK3B (0.69) GSK3BGSK3AAAK1CYP1A2
SCHEMBL4494393 0.88 GSK3B (0.68) GSK3BGSK3AAAK1HDAC6
SCHEMBL4502197 0.87 AAK1 (0.64) GSK3BGSK3AAAK1CYP1A2HDAC6
SCHEMBL4499436 0.86 HDAC6 (0.66) GSK3BGSK3AAAK1HDAC6
SCHEMBL4482990 0.85 GSK3B (0.65) GSK3BGSK3AAAK1CYP1A2HDAC6
SCHEMBL4485505 0.85 GSK3B (0.59) GSK3BGSK3AAAK1CYP1A2HDAC6
SCHEMBL4494613 0.84 GSK3B (0.57) GSK3BGSK3AAAK1CYP1A2HDAC6
SCHEMBL4481457 0.84 GSK3B (0.69) GSK3BGSK3AAAK1CYP1A2HDAC6
SCHEMBL4503079 0.84 HDAC6 (0.69) AAK1HDAC6
SCHEMBL4493555 0.83 AAK1 (0.60) GSK3BGSK3AAAK1CYP1A2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7632854-B2 Aminoindazole derivatives active as kinase inhibitors, process for their preparation and pharmaceutical compositions comprising them PFIZER ITALIA S.R.L. (IT) 2009-12-15 US claimed