SCHEMBL4497716

SCHEMBL4497716

COc1cccc(-c2[nH]c(C=O)c(C(=O)O)c2C(C)C)n1

nearest known ligand 0.41

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
BTK Q06187 2/20 0.41
NR4A2 P43354 1/20 0.33
DHODH Q02127 1/20 0.33
PTGES O14684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4496742 0.85 CCR1 (0.36)
SCHEMBL4492959 0.75 CA12 (0.41) PTGES
SCHEMBL4491011 0.75 SMN1; SMN2 (0.44)
SCHEMBL4488177 0.74 BTK (0.41) BTKPTGES
SCHEMBL4504198 0.72 LDHA (0.38)
SCHEMBL4495798 0.72 ERN1 (0.46)
SCHEMBL4498684 0.72 CSNK1D (0.44)
SCHEMBL4488655 0.70 KDM4E (0.36)
SCHEMBL4491755 0.70 TRPV1 (0.36) DHODH
SCHEMBL4492341 0.67 LDHA (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7504429-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2009-03-17 US claimed