SCHEMBL4510215

SCHEMBL4510215

CC(C)(C)[Si](C)(C)OCc1ccc(NC(=O)O)nc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DEGS1 O15121 3/20 0.42
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
RAB9A P51151 5/20 0.39
MAPT P10636 3/20 0.39
RET P07949 1/20 0.39
NPC1 O15118 4/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
KDM4E B2RXH2 2/20 0.38
LMNA P02545 2/20 0.38
ALDH1A1 P00352 1/20 0.38
TSHR P16473 2/20 0.36
HPGD P15428 1/20 0.36
CASP1 P29466 1/20 0.36
HSD17B10 Q99714 1/20 0.36
USP14 P54578 1/20 0.35
PAX8 Q06710 1/20 0.35
KLF5 Q13887 1/20 0.35
BACE1 P56817 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30643687 0.87 RAB9A (0.38) DEGS1MEN1KMT2ARAB9AMAPT
SCHEMBL14659571 0.84 RAB9A (0.41) DEGS1MEN1KMT2ARAB9AMAPT
SCHEMBL19306519 0.80 KLK7 (0.41) MEN1KMT2ARAB9ANPC1SMN1; SMN2
SCHEMBL15835798 0.79 P4HTM (0.51) MEN1KMT2AMAPTKDM4ELMNA
SCHEMBL101243 0.78 LMNA (0.41) MEN1KMT2ARAB9AMAPTNPC1
SCHEMBL3662587 0.78 CYP11B1 (0.48)
SCHEMBL15620009 0.77 MAPK1 (0.49) RAB9ANPC1KDM4EALDH1A1BACE1
SCHEMBL5743568 0.76 KMT2A (0.34) MEN1KMT2ARAB9AMAPTNPC1
SCHEMBL1535653 0.76 TSHR (0.36) MEN1KMT2ASMN1; SMN2LMNATSHR
SCHEMBL15835799 0.76 P4HTM (0.37) MEN1KMT2ARAB9AMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090325956-A1 Aromatic amine derivative and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-12-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090325956-A1 Aromatic amine derivative and use thereof SCD, SCD5, SMS DEGS1 972/4885MEN1 4180/4885KMT2A 1109/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.