SCHEMBL4512654

SCHEMBL4512654

CC(=O)NCCc1c[nH]c2ccc(F)cc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 7/20 1.00
MTNR1B P49286 7/20 1.00
NOTUM Q6P988 4/20 1.00
CYP1A2 P05177 4/20 0.74
BLM P54132 3/20 0.74
SPR P35270 2/20 0.74
KDM4E B2RXH2 2/20 0.74
ALDH1A1 P00352 2/20 0.74
CYP3A4 P08684 2/20 0.74
CYP2D6 P10635 2/20 0.74
HPGD P15428 2/20 0.74
MAPT P10636 1/20 0.74
IDO1 P14902 1/20 0.74
NPSR1 Q6W5P4 1/20 0.74
MPO P05164 7/20 0.69
NQO2 P16083 3/20 0.69
MEN1 O00255 2/20 0.69
KMT2A Q03164 2/20 0.69
HTR2B P41595 2/20 0.69
CYP1A1 P04798 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4488812 0.89 MTNR1A (0.81) MTNR1AMTNR1BNOTUMCYP1A2BLM
SCHEMBL20242784 0.88 NOTUM (0.78) MTNR1AMTNR1BNOTUMSPRMPO
SCHEMBL2410324 0.87 NOTUM (0.77) MTNR1AMTNR1BNOTUMSPRMPO
SCHEMBL1771902 0.85 MTNR1A (1.00) MTNR1AMTNR1BNOTUMCYP1A2BLM
SCHEMBL31543697 0.85 MTNR1A (1.00) MTNR1AMTNR1BNOTUMCYP1A2BLM
Acetylserotonin SCHEMBL30295379 0.85 SPR (1.00) MTNR1AMTNR1BNOTUMCYP1A2BLM
Acetylserotonin SCHEMBL29375184 0.85 SPR (1.00) MTNR1AMTNR1BNOTUMCYP1A2BLM
Acetylserotonin SCHEMBL422165 0.85 SPR (1.00) MTNR1AMTNR1BNOTUMCYP1A2BLM
SCHEMBL14077525 0.84 NOTUM (0.72) MTNR1AMTNR1BNOTUMCYP1A2BLM
SCHEMBL32678263 0.84 NOTUM (0.77) MTNR1AMTNR1BNOTUMSPRMPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4381284-B1 LIGAND-TARGET INTERACTION ANALYSIS BY PHOTOCHEMICALLY INDUCED DYNAMIC NUCLEAR POLARIZATION (PHOTO-CIDNP) ENHANCED NMR SPECTROSCOPY ETH ZUERICH (CH) 2025-07-09 EP disclosed
WO-2025099444-A1 N-Acetylserotonin (NAS) Analogues Beckley Psytech Limited (GB) 2025-05-15 WO disclosed
US-20240345008-A1 LIGAND-TARGET INTERACTION ANALYSIS BY PHOTOCHEMICALLY INDUCED DYNAMIC NUCLEAR POLARIZATION (PHOTO-CIDNP) ENHANCED NMR SPECTROSCOPY ETH ZURICH (CH) 2024-10-17 US disclosed
EP-4381284-A1 LIGAND-TARGET INTERACTION ANALYSIS BY PHOTOCHEMICALLY INDUCED DYNAMIC NUCLEAR POLARIZATION (PHOTO-CIDNP) ENHANCED NMR SPECTROSCOPY ETH Zurich (CH) 2024-06-12 EP disclosed
WO-2023012203-A1 LIGAND-TARGET INTERACTION ANALYSIS BY PHOTOCHEMICALLY INDUCED DYNAMIC NUCLEAR POLARIZATION (PHOTO-CIDNP) ENHANCED NMR SPECTROSCOPY ETH ZURICH (CH) 2023-02-09 WO disclosed
EP-4130727-A1 LIGAND-TARGET INTERACTION ANALYSIS BY PHOTOCHEMICALLY INDUCED DYNAMIC NUCLEAR POLARIZATION (PHOTO-CIDNP) ENHANCED NMR SPECTROSCOPY ETH Zurich (CH) 2023-02-08 EP disclosed
US-20190247527-A1 18F-Labeled Compounds for PET Imaging and Uses Thereof THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL 2019-08-15 US disclosed
US-7612099-B2 Vinylogous acid derivatives HOFFMANN-LA ROCHE INC. (US) 2009-11-03 US disclosed
CN-101321749-A Novel vinylogous acid derivatives HOFFMANN LA ROCHE (CH) 2008-12-10 CN disclosed
EP-1957483-A1 NOVEL VINYLOGOUS ACIDS DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2008-08-20 EP disclosed
WO-2007063010-A1 NOVEL VINYLOGOUS ACIDS DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2007-06-07 WO disclosed
US-20070129421-A1 Vinylogous acid derivatives HOFFMANN-LA ROCHE INC. 2007-06-07 US disclosed
WO-2004085392-A1 MELATONIN DERIVATIVES AND THEIR USE FOR TREATING NEUROLOGICAL DYSFUNCTIONS FAUST PHARMACEUTICALS (FR) 2004-10-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190247527-A1 18F-Labeled Compounds for PET Imaging and Uses Thereof IDO1, IDO2, CD274 MTNR1A 1167/4885MTNR1B 1523/4885NOTUM 2973/4885
US-20070129421-A1 Vinylogous acid derivatives CMA1, TPSG1, TPSAB1 MTNR1A 454/4885MTNR1B 756/4885NOTUM 601/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.