SCHEMBL4517205

SCHEMBL4517205

CC(=O)OC(C=O)Cc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.46
ALPI P09923 1/20 0.46
PKM P14618 1/20 0.46
PTGS1 P23219 1/20 0.46
XIAP P98170 1/20 0.46
SLC7A5 Q01650 1/20 0.46
CYP1A2 P05177 1/20 0.44
CTSK P43235 6/20 0.44
CTSL P07711 3/20 0.44
CTSB P07858 3/20 0.44
CTSH P09668 2/20 0.44
SRR Q9GZT4 2/20 0.42
TSHR P16473 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
TAAR1 Q96RJ0 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
CTRB1 P17538 2/20 0.41
ALPL P05186 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27580730 1.00 ALDH1A1 (0.46) ALDH1A1ALPIPKMPTGS1XIAP
SCHEMBL13223447 0.86 CYP1A2 (0.47) ALPIPKMPTGS1XIAPSLC7A5
SCHEMBL10404341 0.85 ALDH1A1 (0.44) ALDH1A1ALPIPKMPTGS1XIAP
SCHEMBL8376755 0.85 ALDH1A1 (0.44) ALDH1A1ALPIPKMPTGS1XIAP
SCHEMBL14297463 0.84 ALPI (0.41) ALDH1A1ALPIPKMPTGS1XIAP
SCHEMBL11110716 0.83 MMP12 (0.50) ALDH1A1CYP1A2CTSKTSHRMEN1
SCHEMBL28540100 0.83 SRR (0.46) ALPIPKMPTGS1XIAPSLC7A5
SCHEMBL7296959 0.83 SRR (0.46) ALPIPKMPTGS1XIAPSLC7A5
SCHEMBL14762630 0.83 SRR (0.46) ALPIPKMPTGS1XIAPSLC7A5
SCHEMBL678123 0.82 CTSK (0.41) ALPIPKMPTGS1XIAPSLC7A5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-4294903-B2 2009-07-15 JP claimed
JP-2003519135-A 2003-06-17 JP claimed
EP-1242400-A1 PYRROLIDINE DERIVATIVES AS CYCLIC AMP-SPECIFIC PHOSPHODIESTERASE INHIBITORS ICOS CORPORATION (US) 2002-09-25 EP claimed
WO-2001047905-A1 PYRROLIDINE DERIVATIVES AS CYCLIC AMP-SPECIFIC PHOSPHODIESTERASE INHIBITORS ICOS CORPORATION (US) 2001-07-05 WO claimed
EP-0184550-B1 5-AMINO-4-HYDROXY VALERYL AMIDE DERIVATIVES CIBA-GEIGY AG (CH) 1992-03-18 EP disclosed
US-4931591-A Novel 5-amino-4-hydroxyvaleryl derivatives CIBA-GEIGY CORPORATION (US) 1990-06-05 US disclosed
US-4727060-A HYPOTENSIVE AGENTS CIBA-GEIGY CORPORATION (US) 1988-02-23 US disclosed
EP-0184550-A2 5-Amino-4-hydroxy valeryl amide derivatives CIBA-GEIGY AG (CH) 1986-06-11 EP disclosed
EP-0126849-A1 Pharmacologically active N-amino hydantoin derivatives, their synthesis and intermediates THE WELLCOME FOUNDATION LIMITED (GB) 1984-12-05 EP disclosed