SCHEMBL4527092

SCHEMBL4527092

CCOc1ccccc1-n1c(CC)nc2c(cnn2-c2ccccc2)c1=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.58
TP53 P04637 1/20 0.58
MAPT P10636 2/20 0.54
DPP4 P27487 5/20 0.54
LMNA P02545 3/20 0.53
TSHR P16473 3/20 0.53
HTT P42858 2/20 0.53
XBP1 P17861 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.52
POLB P06746 2/20 0.52
GRM1 Q13255 3/20 0.51
GRM5 P41594 1/20 0.50
CSNK2A2 P19784 1/20 0.50
CSNK2B P67870 1/20 0.50
CSNK2A1 P68400 1/20 0.50
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 1/20 0.48
HPGD P15428 1/20 0.48
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4528163 0.85 HIF1A (0.71) SMN1; SMN2DPP4LMNATSHRNPSR1
SCHEMBL13789635 0.84 DPP4 (0.47) SMN1; SMN2MAPTDPP4LMNATSHR
SCHEMBL4465299 0.79 L3MBTL1 (0.79) SMN1; SMN2LMNATSHRNPSR1L3MBTL1
SCHEMBL13789510 0.79 HIF1A (0.51) SMN1; SMN2DPP4LMNATSHRHTT
SCHEMBL4507484 0.77 L3MBTL1 (0.61) SMN1; SMN2LMNATSHRNPSR1L3MBTL1
SCHEMBL13789634 0.75 L3MBTL1 (0.58) SMN1; SMN2LMNATSHRNPSR1L3MBTL1
SCHEMBL2116934 0.74 NPSR1 (0.67) SMN1; SMN2TP53MAPTDPP4LMNA
SCHEMBL2118435 0.72 MAPT (0.73) SMN1; SMN2TP53MAPTLMNATSHR
SCHEMBL939933 0.72 ALDH1A1 (0.64) SMN1; SMN2TP53LMNATSHRHTT
SCHEMBL1592824 0.72 L3MBTL1 (0.60) SMN1; SMN2MAPTLMNATSHRNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090170834-A1 Fused Pyrimidones and Thiopyrimidones, and Uses Thereof PROLEXYS PHARMACEUTICALS, INC. (US) 2009-07-02 US disclosed
US-20090170834-A1 Fused Pyrimidones and Thiopyrimidones, and Uses Thereof PROLEXYS PHARMACEUTICALS, INC. (US) 2009-07-02 US disclosed
US-20090170834-A1 Fused Pyrimidones and Thiopyrimidones, and Uses Thereof PROLEXYS PHARMACEUTICALS, INC. (US) 2009-07-02 US disclosed
WO-2007076085-A2 FUSED PYRIMIDONES AND THIOPYRIMIDONES, AND USES THEREOF PROLEXYS PHARMACEUTICALS, INC . (US) 2007-07-05 WO disclosed
WO-2007076085-A2 FUSED PYRIMIDONES AND THIOPYRIMIDONES, AND USES THEREOF PROLEXYS PHARMACEUTICALS, INC . (US) 2007-07-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090170834-A1 Fused Pyrimidones and Thiopyrimidones, and Uses Thereof TYMP, TYMS, MKI67 SMN1; SMN2 1145/4885TP53 47/4885MAPT 4007/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.