SCHEMBL4527646

SCHEMBL4527646

Cc1ccnc2c1c(C(=O)NCC1(N3CCN[C@@H](C)C3)CCCCC1)cn2-c1ncccn1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HCN4 Q9Y3Q4 14/20 0.42
HCN1 O60741 11/20 0.42
HCN3 Q9P1Z3 1/20 0.42
HCN2 Q9UL51 1/20 0.42
ALDH1A1 P00352 1/20 0.41
TSHR P16473 1/20 0.41
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
GAA P10253 1/20 0.38
TP53 P04637 1/20 0.37
THRB P10828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4540375 0.89 HCN1 (0.44) HCN4HCN1HCN3HCN2ALDH1A1
SCHEMBL13706601 0.89 HCN1 (0.44) HCN4HCN1HCN3HCN2ALDH1A1
SCHEMBL13706853 0.85 HCN1 (0.60) HCN4HCN1ALDH1A1TSHRMEN1
SCHEMBL13706969 0.85 HCN1 (0.41) HCN4HCN1HCN3HCN2ALDH1A1
SCHEMBL13706894 0.84 ALDH1A1 (0.58) HCN4HCN1ALDH1A1TSHRTHRB
SCHEMBL13706876 0.84 HCN4 (0.39) HCN4HCN1HCN3HCN2ALDH1A1
SCHEMBL13706774 0.84 HCN4 (0.55) HCN4HCN1HCN3HCN2ALDH1A1
SCHEMBL4364179 0.83 P2RX7 (0.48) HCN4HCN1HCN3HCN2ALDH1A1
SCHEMBL13706815 0.83 P2RX7 (0.48) HCN4HCN1HCN3HCN2ALDH1A1
SCHEMBL4358058 0.83 HCN1 (0.42) HCN4HCN1HCN3HCN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009108551-A2 HETEROARYL AMIDE ANALOGUES H. LUNDBECK A/S (DK) 2009-09-03 WO claimed
WO-2009108551-A2 HETEROARYL AMIDE ANALOGUES H. LUNDBECK A/S (DK) 2009-09-03 WO disclosed