SCHEMBL4532945

SCHEMBL4532945

Cc1onc2cc(O)ccc12

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 1/20 0.45
ESR1 P03372 8/20 0.45
ESR2 Q92731 8/20 0.45
HSP90AA1 P07900 1/20 0.41
HSP90AB1 P08238 1/20 0.41
DYRK1A Q13627 1/20 0.40
ALDH1A1 P00352 3/20 0.39
HSD17B10 Q99714 3/20 0.39
ALOX15 P16050 2/20 0.39
KDM4E B2RXH2 2/20 0.39
LMNA P02545 2/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
GAA P10253 2/20 0.39
HPGD P15428 2/20 0.39
CASP1 P29466 2/20 0.39
CASP7 P55210 2/20 0.39
TSHR P16473 1/20 0.39
HSD17B3 P37058 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19555431 0.84 DYRK1A (0.51) ENPP2ESR1ESR2HSP90AA1HSP90AB1
SCHEMBL16431700 0.79 ENPP2 (0.48) ENPP2ESR1ESR2HSP90AA1ALDH1A1
SCHEMBL8404501 0.79 DYRK1A (0.42) DYRK1AALDH1A1HSD17B10KDM4ELMNA
SCHEMBL21596940 0.76 ENPP2 (0.45) ENPP2ESR1ESR2HSP90AA1ALDH1A1
SCHEMBL18822704 0.76 DYRK1A (0.40) DYRK1A
SCHEMBL14353775 0.76 MPO (0.41) DYRK1AALDH1A1ALOX15KDM4ELMNA
SCHEMBL24943958 0.73 DYRK1A (0.38) DYRK1AALDH1A1HSD17B10ALOX15LMNA
SCHEMBL6818471 0.72 ENPP2 (0.41) ENPP2ESR1ESR2HSP90AA1ALDH1A1
SCHEMBL17437927 0.71 CA12 (0.44) ENPP2ESR2ALDH1A1HSD17B10KDM4E
SCHEMBL1423001 0.70 GPR3 (0.46) DYRK1AALDH1A1HSD17B10ALOX15LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2638008-A1 LACTAM DERIVATIVES USEFUL AS OREXIN RECEPTOR ANTAGONISTS Actelion Pharmaceuticals Ltd. (CH) 2013-09-18 EP disclosed
WO-2012063207-A1 LACTAM DERIVATIVES USEFUL AS OREXIN RECEPTOR ANTAGONISTS ACTELION PHARMACEUTICALS LTD (CH) 2012-05-18 WO disclosed