SCHEMBL4533110

SCHEMBL4533110

Cc1ccccc1S(=O)(=O)N1CCC(CNC(=O)C23CC4CC(CC(C4)C2)C3)C1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.46
EPHX2 P34913 3/20 0.44
P2RX7 Q99572 1/20 0.43
ALDH1A1 P00352 2/20 0.42
CACNA1H O95180 1/20 0.41
LMNA P02545 2/20 0.41
GAA P10253 2/20 0.41
HSD11B1 P28845 1/20 0.41
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
POLB P06746 1/20 0.40
CCR1 P32246 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4542865 0.95 HPGD (0.43) HPGDEPHX2P2RX7ALDH1A1CACNA1H
SCHEMBL4533158 0.94 EPHX2 (0.48) HPGDEPHX2P2RX7ALDH1A1CACNA1H
SCHEMBL8064823 0.88 HPGD (0.46) HPGDEPHX2P2RX7ALDH1A1CACNA1H
SCHEMBL4539753 0.88 HDAC3 (0.49) HPGDEPHX2P2RX7ALDH1A1LMNA
SCHEMBL8049830 0.86 HSD11B1 (0.49) HSD11B1
SCHEMBL4539563 0.86 EPHX2 (0.56) EPHX2
SCHEMBL4539749 0.86 HSD11B1 (0.45) HPGDALDH1A1LMNAGAAHSD11B1
SCHEMBL4542831 0.85 ALDH1A1 (0.53) HPGDEPHX2ALDH1A1LMNAGAA
SCHEMBL4532816 0.83 TP53 (0.48) ALDH1A1LMNAGAAPOLB
SCHEMBL4538127 0.83 CCR1 (0.46) HPGDEPHX2P2RX7HSD11B1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed