SCHEMBL4534329

SCHEMBL4534329

COc1cccc(S(=O)(=O)N2CCC(CNC(=O)C34CC5CC(CC(C5)C3)C4)C2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 5/20 0.49
CHRM5 P08912 1/20 0.45
P2RX2 Q9UBL9 1/20 0.45
POLB P06746 3/20 0.45
ALDH1A1 P00352 3/20 0.45
LMNA P02545 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
HPGD P15428 1/20 0.45
HSD17B10 Q99714 1/20 0.45
USP2 O75604 1/20 0.45
KMT2A Q03164 3/20 0.44
NPC1 O15118 1/20 0.44
APOBEC3A P31941 1/20 0.44
APOBEC3G Q9HC16 1/20 0.44
MAPT P10636 3/20 0.44
MEN1 O00255 1/20 0.43
MCL1 Q07820 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
THRB P10828 1/20 0.43
USP5 P45974 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8060988 1.00 PKM (0.49) PKMCHRM5P2RX2POLBALDH1A1
SCHEMBL8048322 0.88 ALDH1A1 (0.45) PKMPOLBALDH1A1LMNAHPGD
SCHEMBL4530583 0.88 EPHX2 (0.46) POLBALDH1A1LMNAHPGDUSP2
SCHEMBL4543002 0.88 ALDH1A1 (0.45) PKMPOLBALDH1A1LMNAHPGD
SCHEMBL4539990 0.87 USP2 (0.56) PKMPOLBALDH1A1LMNAUSP2
SCHEMBL8053633 0.87 ALDH1A1 (0.43) PKMPOLBALDH1A1LMNASMN1; SMN2
SCHEMBL4535853 0.86 FBP1 (0.46) ALDH1A1LMNASMN1; SMN2HPGDKMT2A
SCHEMBL4542831 0.85 ALDH1A1 (0.53) PKMALDH1A1LMNAHPGDKMT2A
SCHEMBL4541158 0.84 ALDH1A1 (0.49) POLBALDH1A1LMNASMN1; SMN2HPGD
SCHEMBL4541786 0.84 NPC1 (0.55) POLBALDH1A1LMNASMN1; SMN2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed