SCHEMBL4536909

SCHEMBL4536909

O=C(O)C1=CN=Cc2ccccc2C1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
TRPA1 O75762 9/20 0.41
SRD5A2 P31213 2/20 0.33
MTNR1A P48039 1/20 0.31
MTNR1B P49286 1/20 0.31
GSR P00390 1/20 0.31
DAO P14920 1/20 0.30
TSHR P16473 1/20 0.30
NAPRT Q6XQN6 1/20 0.30
ALDH1A1 P00352 1/20 0.30
ALOX15 P16050 1/20 0.30
SRD5A1 P18405 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL8881145 0.91 MAOA (0.38) MAOAMAOBTRPA1
SCHEMBL29906826 0.76 MAOA (0.59) MAOAMAOBTRPA1SRD5A2MTNR1A
SCHEMBL1067727 0.76 MAOA (0.59) MAOAMAOBTRPA1SRD5A2MTNR1A
SCHEMBL7334826 0.76 TRPA1 (0.38) MAOAMAOBTRPA1TSHR
SCHEMBL5026786 0.74 TRPA1 (0.46) MAOAMAOBTRPA1
SCHEMBL20613152 0.74 TRPA1 (0.48) MAOAMAOBTRPA1TSHR
SCHEMBL6273946 0.73 MAOA (0.47) MAOAMAOBTRPA1SRD5A2MTNR1A
SCHEMBL7500741 0.72 MAOA (0.44) MAOAMAOBTRPA1SRD5A2MTNR1A
SCHEMBL27562448 0.71 MAOA (0.46) MAOAMAOBTRPA1SRD5A2MTNR1A
Biphenyl SCHEMBL27655126 0.71 MAOA (0.59) MAOAMAOBTRPA1SRD5A2MTNR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2638017-A1 CRYSTALLINE FORMS OF AN ALKOXYIMIDAZOL-1-YLMETHYL BIPHENYL CARBOXYLIC ACID Theravance, Inc. (US) 2013-09-18 EP disclosed
WO-2012064807-A1 CRYSTALLINE FORMS OF AN ALKOXYIMIDAZOL-1-YLMETHYL BIPHENYL CARBOXYLIC ACID THERAVANCE, INC. (US) 2012-05-18 WO disclosed
US-5679671-A ANGIOTENSIN 1-CONVERTING ENZYME INHIBITOR, VASOPRESSIN ANTAGONISM AND ATRIAL NAUTRIURETIC PEPTIDE HYDROLASE INHIBITOR EISAI CO., LTD. (JP) 1997-10-21 US disclosed
US-5529995-A Aminoacetylmercapto derivatives useful as inhibitors of enkephalinase and ACE MERRELL DOW PHARMACEUTICALS INC. (US) 1996-06-25 US disclosed