SCHEMBL5026786

SCHEMBL5026786

OC1=CN=Cc2ccccc2C1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 9/20 0.46
MAOA P21397 1/20 0.33
MAOB P27338 1/20 0.33
CYP11B2 P19099 2/20 0.32
CYP11B1 P15538 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20613152 0.79 TRPA1 (0.48) TRPA1MAOAMAOBCYP11B2CYP11B1
SCHEMBL4536909 0.74 MAOA (0.44) TRPA1MAOAMAOB
SCHEMBL275380 0.72 MAOA (0.47) TRPA1MAOAMAOBCYP11B2CYP11B1
SCHEMBL7334826 0.71 TRPA1 (0.38) TRPA1MAOAMAOB
Trifluoroacetic Acid SCHEMBL8881145 0.68 MAOA (0.38) TRPA1MAOAMAOB
SCHEMBL2713020 0.67 PARP1 (0.36) TRPA1MAOAMAOBCYP11B2CYP11B1
SCHEMBL3101816 0.66 TRPA1 (0.42) TRPA1CYP11B2
SCHEMBL7436002 0.64 TRPA1 (0.42) TRPA1MAOAMAOBCYP11B2
SCHEMBL6997599 0.64 TRPA1 (0.46) TRPA1MAOAMAOBCYP11B2CYP11B1
SCHEMBL3707900 0.64 TRPA1 (0.46) TRPA1MAOAMAOBCYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904069-A2 ARYL-AND HETEROARYL-SUBSTITUTED TETRAHYDROBENZAZEPINES AND USE THEREOF TO BLOCK REUPTAKE OF NOREPINEPHRINE, DOPAMINE, AND SEROTONIN AMR Technology, Inc. (US) 2008-04-02 EP disclosed
WO-2007011820-A2 ARYL-AND HETEROARYL-SUBSTITUTED TETRAHYDROBENZAZEPINES AND USE THEREOF TO BLOCK REUPTAKE OF NOREPINEPHRINE, DOPAMINE, AND SEROTONIN AMR TECHNOLOGY, INC. (US) 2007-01-25 WO disclosed