SCHEMBL4537075

SCHEMBL4537075

COc1ccc(S(=O)(=O)N2CCCC(CNC(=O)NC34CC5CC(CC(C5)C3)C4)C2)c(OC)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.53
KMT2A Q03164 3/20 0.49
MEN1 O00255 2/20 0.49
LMNA P02545 2/20 0.49
HTT P42858 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
EPHX1 P07099 9/20 0.48
EPHX2 P34913 8/20 0.48
POLB P06746 1/20 0.47
ALDH1A1 P00352 2/20 0.46
NPSR1 Q6W5P4 2/20 0.46
KDM4E B2RXH2 1/20 0.46
USP2 O75604 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
MAPT P10636 1/20 0.46
CYP2C9 P11712 1/20 0.46
ALOX15 P16050 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4536597 0.88 CYP19A1 (0.54) CYP19A1KMT2AMEN1LMNAHTT
SCHEMBL4537586 0.87 EPHX1 (0.52) LMNAHTTEPHX1EPHX2ALDH1A1
SCHEMBL4537010 0.84 EPHX2 (0.55) EPHX1EPHX2
SCHEMBL4541158 0.84 ALDH1A1 (0.49) CYP19A1KMT2AMEN1LMNAHTT
SCHEMBL4538117 0.82 FKBP1A (0.48) KMT2AMEN1LMNASMN1; SMN2EPHX1
SCHEMBL4535739 0.82 EPHX2 (0.54) LMNAEPHX1EPHX2ALDH1A1NPSR1
SCHEMBL4542230 0.81 CYP19A1 (0.54) CYP19A1KMT2AMEN1LMNAHTT
SCHEMBL4535087 0.81 EPHX1 (0.49) LMNAHTTEPHX1EPHX2NPSR1
SCHEMBL4539990 0.81 USP2 (0.56) KMT2AMEN1LMNAEPHX1EPHX2
SCHEMBL8062507 0.81 EPHX2 (0.53) EPHX1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009083526-A1 NOVEL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2009-07-09 WO disclosed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed