SCHEMBL4537586

SCHEMBL4537586

COc1ccc(S(=O)(=O)N2CCCC(CNC(=O)NC34CC5CC(CC(C5)C3)C4)C2)cc1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 9/20 0.52
EPHX2 P34913 9/20 0.52
NPC1 O15118 1/20 0.52
HTT P42858 1/20 0.51
ALDH1A1 P00352 3/20 0.51
LMNA P02545 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
TSHR P16473 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4535739 0.95 EPHX2 (0.54) EPHX1EPHX2ALDH1A1LMNANPSR1
SCHEMBL4542200 0.90 LMNA (0.54) EPHX1EPHX2LMNA
SCHEMBL4540005 0.88 LMNA (0.57) EPHX1EPHX2HTTLMNANPSR1
SCHEMBL4542921 0.88 CYP3A4 (0.57) EPHX1EPHX2NPC1ALDH1A1
SCHEMBL8060768 0.88 LMNA (0.57) EPHX1EPHX2HTTLMNANPSR1
SCHEMBL8062904 0.88 EPHX2 (0.59) EPHX1EPHX2ALDH1A1
SCHEMBL4537319 0.87 ALDH1A1 (0.52) EPHX1NPC1HTTALDH1A1LMNA
SCHEMBL4541786 0.87 NPC1 (0.55) NPC1HTTALDH1A1LMNATSHR
SCHEMBL4537075 0.87 CYP19A1 (0.53) EPHX1EPHX2HTTALDH1A1LMNA
SCHEMBL4541299 0.85 EPHX1 (0.51) EPHX1EPHX2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed