SCHEMBL4537987

SCHEMBL4537987

Cc1cnc(C(CO)N(C)Cc2ccc(Cl)nc2Cl)s1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSA P10619 18/20 0.33
MEN1 O00255 1/20 0.30
NPC1 O15118 1/20 0.30
POLB P06746 1/20 0.30
RAB9A P51151 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3714125 0.79 RAB9A (0.32) CTSAMEN1NPC1POLBRAB9A
SCHEMBL4543601 0.75 AOC3 (0.34)
SCHEMBL4537085 0.72 OPRM1 (0.36)
SCHEMBL4539599 0.67
SCHEMBL3699960 0.65 CHRM1 (0.32)
SCHEMBL4540382 0.63 CTSA (0.39) CTSA
SCHEMBL3700231 0.61 RAB9A (0.34) RAB9A
SCHEMBL30968506 0.60 KDM4E (0.40) NPC1RAB9AKMT2A
SCHEMBL844810 0.60 KDM4E (0.40) NPC1RAB9AKMT2A
SCHEMBL17018453 0.60 NOS1 (0.42) CTSA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064269-A1 COMPOUNDS AND THEIR USE FOR TREATMENT OF Αβ-RELATED DISEASES ASTRAZENECA AB (SE) 2012-05-18 WO disclosed