SCHEMBL4538466

SCHEMBL4538466

CC(C)(C=O)Oc1ccc(C(=O)c2ccc(Cl)cc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 9/20 0.65
PPARG P37231 4/20 0.65
FABP2 P12104 2/20 0.65
SLC22A12 Q96S37 1/20 0.65
ELANE P08246 2/20 0.58
CYP1A2 P05177 3/20 0.57
CYP3A4 P08684 3/20 0.57
MAPT P10636 3/20 0.57
SMN1; SMN2 Q16637 3/20 0.57
HPGD P15428 2/20 0.57
MEN1 O00255 2/20 0.57
CYP2C19 P33261 2/20 0.57
KMT2A Q03164 2/20 0.57
MAPK1 P28482 2/20 0.57
ABCB11 O95342 2/20 0.57
TSHR P16473 2/20 0.57
HTR2A P28223 2/20 0.57
PMP22 Q01453 2/20 0.57
LMNA P02545 2/20 0.57
USP2 O75604 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3496791 0.88 PPARA (0.53) PPARAPPARGFABP2SLC22A12ELANE
SCHEMBL4540353 0.86 PPARA (0.60) PPARAPPARGFABP2SLC22A12ELANE
SCHEMBL4540357 0.86 PPARA (0.60) PPARAPPARGFABP2SLC22A12ELANE
SCHEMBL13198222 0.84 TRPV1 (0.46) PPARAPPARGFABP2SLC22A12ELANE
SCHEMBL10190646 0.83 PPARA (0.73) PPARAPPARGFABP2SLC22A12ELANE
SCHEMBL30657556 0.80 PPARA (0.69) PPARAPPARGFABP2SLC22A12ELANE
SCHEMBL21886332 0.80 CA1 (0.52) PPARAPPARGFABP2SLC22A12SMN1; SMN2
SCHEMBL822492 0.79 PPARA (0.77) PPARAPPARGFABP2SLC22A12ELANE
SCHEMBL13984052 0.79 PPARA (0.77) PPARAPPARGFABP2SLC22A12ELANE
Fenofibric Acid SCHEMBL16377 0.79 PPARA (1.00) PPARAPPARGFABP2SLC22A12ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 27 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240189287-A1 PERIPHERALLY RESTRICTED CB1 RECEPTOR BLOCKERS AND USES THEREOF BIONANOSIM (BNS) LTD (IL) 2024-06-13 US disclosed
CN-107021943-B 7-epi-baccatin III derivatives, and preparation method and application thereof 中国科学院上海药物研究所 2020-12-29 CN disclosed
WO-2020146876-A2 ANTI-CANCER COMPOSITIONS AND METHODS OF USE BOARD OF SUPERVISORS OF LOUISIANA STATE UNIVERSITY AND AGRICULTURAL AND MECHANICAL COLLEGE (US) 2020-07-16 WO disclosed
US-8946224-B2 Substituted [1,2,4]triazolo[4,3-A]pyrazines for medicaments and pharmaceutical compositions REDX PHARMA LIMITED (GB) 2015-02-03 US disclosed
US-8946224-B2 Substituted [1,2,4]triazolo[4,3-A]pyrazines for medicaments and pharmaceutical compositions REDX PHARMA LIMITED (GB) 2015-02-03 US disclosed
US-8946224-B2 Substituted [1,2,4]triazolo[4,3-A]pyrazines for medicaments and pharmaceutical compositions REDX PHARMA LIMITED (GB) 2015-02-03 US disclosed
EP-2638007-A2 DRUG DERIVATIVES Redx Pharma Limited (GB) 2013-09-18 EP disclosed
US-20130225594-A1 DRUG DERIVATIVES REDX PHARMA PLC (GB) 2013-08-29 US disclosed
US-20130225594-A1 DRUG DERIVATIVES REDX PHARMA PLC (GB) 2013-08-29 US disclosed
US-20130225594-A1 DRUG DERIVATIVES REDX PHARMA PLC (GB) 2013-08-29 US disclosed
US-20050037997-A9 Materials and methods for the treatment of diabetes, hyperlipidemia, hypercholesterolemia, and atherosclerosis MPM ASSET MANAGEMENT INVESTORS 2002 BVIII LLC 2005-02-17 US disclosed
US-6768008-B2 FOR THERAPY ARYX THERAPEUTICS 2004-07-27 US disclosed
EP-1430039-A2 ARYL DERIVATIVES FOR THE TREATMENT OF DIABETES, HYPERLIPIDEMIA, HYPERCHOLESTEROLEMIA AND ATHEROSCLEROSIS Aryx Therapeutics (US) 2004-06-23 EP disclosed
US-6680387-B2 USING THIAZOLIDINONE COMPOUND ARYX THERAPEUTICS 2004-01-20 US disclosed
US-20030236227-A1 Materials and methods for the treatment of diabetes, hyperlipidemia, hypercholesterolemia, and atherosclerosis ARYX THERAPEUTICS 2003-12-25 US disclosed
US-20030064972-A1 Materials and methods for the treatment of diabetes, hyperlipidemia, hypercholesterolemia, and atherosclerosis MPM ASSET MANAGEMENT INVESTORS 2002 BVIII LLC 2003-04-03 US disclosed
WO-2003024943-A2 ARYL DERIVATIVES FOR THE TREATMENT OF DIABETES, HYPERLIPIDEMIA, HYPERCHOLESTEROLEMIA AND ATHEROSCLEROSIS ARYX THERAPEUTICS (US) 2003-03-27 WO disclosed
US-20030027798-A1 Materials and methods for the treatment of diabetes, hyperlipidemia, hypercholesterolemia, and atherosclerosis MPM ASSET MANAGEMENT INVESTORS 2002 BVIII LLC 2003-02-06 US disclosed
EP-1276730-A2 THIAZOLIDINEDIONE ANALOGUES AND THEIR USE FOR THE TREATMENT OF DIABETES ARYx Therapeutics (US) 2003-01-22 EP disclosed
WO-2001081328-A2 THIAZOLIDINEDIONE ANALOGUES AND THEIR USE FOR THE TREATMENT OF DIABETES ARYX THERAPEUTICS (US) 2001-11-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030236227-A1 Materials and methods for the treatment of diabetes, hyperlipidemia, hypercholesterolemia, and atherosclerosis LIPA, LIPC, CETP PPARA 305/4885PPARG 370/4885FABP2 258/4885
US-20130225594-A1 DRUG DERIVATIVES SQOR, NQO1, CYP2D6 PPARA 1494/4885PPARG 1203/4885FABP2 4580/4885
US-20030064972-A1 Materials and methods for the treatment of diabetes, hyperlipidemia, hypercholesterolemia, and atherosclerosis LIPA, LIPC, CETP PPARA 305/4885PPARG 370/4885FABP2 258/4885
US-20240189287-A1 PERIPHERALLY RESTRICTED CB1 RECEPTOR BLOCKERS AND USES THEREOF CNR1, CNR2, GPR18 PPARA 241/4885PPARG 209/4885FABP2 294/4885
US-20030027798-A1 Materials and methods for the treatment of diabetes, hyperlipidemia, hypercholesterolemia, and atherosclerosis LIPA, LIPC, CETP PPARA 305/4885PPARG 370/4885FABP2 258/4885
US-20050037997-A9 Materials and methods for the treatment of diabetes, hyperlipidemia, hypercholesterolemia, and atherosclerosis LIPA, LIPC, CETP PPARA 305/4885PPARG 370/4885FABP2 258/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.