SCHEMBL4539667

SCHEMBL4539667

O=C(O)Cc1ccc(N2CCN(Cc3ccccc3)CC2)cc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 5/20 0.71
ITGA2B P08514 5/20 0.71
DRD4 P21917 3/20 0.68
HTR2A P28223 1/20 0.63
HTR2C P28335 1/20 0.63
HTR2B P41595 1/20 0.63
HTR7 P34969 2/20 0.59
HDAC3 O15379 1/20 0.55
HDAC4 P56524 1/20 0.55
HDAC1 Q13547 1/20 0.55
HDAC7 Q8WUI4 1/20 0.55
HDAC2 Q92769 1/20 0.55
HDAC10 Q969S8 1/20 0.55
HDAC11 Q96DB2 1/20 0.55
HDAC8 Q9BY41 1/20 0.55
HDAC6 Q9UBN7 1/20 0.55
HDAC9 Q9UKV0 1/20 0.55
HDAC5 Q9UQL6 1/20 0.55
DRD2 P14416 1/20 0.55
DRD3 P35462 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8691440 0.95 DRD4 (0.70) ITGB3ITGA2BDRD4HTR2AHTR2C
Hydrochloric Acid SCHEMBL8690310 0.94 DRD4 (0.68) ITGB3ITGA2BDRD4HTR2AHTR2C
SCHEMBL10901064 0.90 ITGB3 (0.70) ITGB3ITGA2BDRD4HTR7DRD2
SCHEMBL7364364 0.85 DRD4 (0.59) ITGB3ITGA2BDRD4HTR2AHTR2C
SCHEMBL8744975 0.85 ITGB3 (0.64) ITGB3ITGA2BDRD4ALDH1A1SIGMAR1
SCHEMBL1066467 0.83 HTR2A (0.72) ITGB3ITGA2BDRD4HTR2AHTR2C
SCHEMBL3320211 0.83 DRD4 (0.74) DRD4HTR2AHTR2CHTR2BHTR7
SCHEMBL10900437 0.82 ADRA1D (0.62) HDAC4HDAC1DRD2LMNAALDH1A1
SCHEMBL7459360 0.82 HTR2A (0.71) ITGB3ITGA2BDRD4HTR2AHTR2C
Hydrochloric Acid SCHEMBL4653252 0.82 HTR2A (0.71) ITGB3ITGA2BDRD4HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064569-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-05-18 WO disclosed
EP-0858453-A1 5-(ACETAMIDOMETHYL)-3-ARYLDIHYDROFURAN-2-ONE AND TETRAHYDROFURAN-2-ONE DERIVATIVES WITH ANTIBIOTIC ACTIVITY AstraZeneca AB (SE) 1998-08-19 EP disclosed
WO-1997014690-A1 5-(ACETAMIDOMETHYL)-3-ARYLDIHYDROFURAN-2-ONE AND TETRAHYDROFURAN-2-ONE DERIVATIVES WITH ANTIBIOTIC ACTIVITY ZENECA LIMITED (GB) 1997-04-24 WO disclosed