SCHEMBL4540580

SCHEMBL4540580

CCNc1nc(NC(C)=O)ccc1C(N)=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 4/20 0.50
PGK1 P00558 2/20 0.43
ALDH1A1 P00352 2/20 0.41
HSD17B10 Q99714 2/20 0.41
KDM4E B2RXH2 2/20 0.41
HPGD P15428 1/20 0.41
PARP1 P09874 2/20 0.40
DHODH Q02127 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
SYK P43405 1/20 0.40
PTK2 Q05397 2/20 0.40
LMNA P02545 1/20 0.40
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
MAPK9 P45984 1/20 0.36
MAPT P10636 1/20 0.36
SCN9A Q15858 1/20 0.36
SCN2A Q99250 1/20 0.36
SCN3A Q9NY46 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23009954 0.78 KDM4E (0.43) MAPK8PGK1ALDH1A1HSD17B10KDM4E
SCHEMBL3569662 0.78 PARP1 (0.55) MAPK8PGK1ALDH1A1HSD17B10KDM4E
SCHEMBL2122993 0.70 ALDH1A1 (0.77) ALDH1A1HSD17B10KDM4EHPGDPARP1
SCHEMBL912928 0.69 EGFR (0.59) MAPK8SYKMAPK9
SCHEMBL28477220 0.68 NNMT (0.47) ALDH1A1HSD17B10PARP1
SCHEMBL4540577 0.68 PGK1 (0.44) MAPK8PGK1ALDH1A1HSD17B10KDM4E
SCHEMBL7092192 0.67 SMN1; SMN2 (0.48) MAPK8ALDH1A1HSD17B10KDM4EPTK2
SCHEMBL9143700 0.67 KDM4E (0.46) MAPK8ALDH1A1HSD17B10KDM4EKMT2A
SCHEMBL2627049 0.67 SYK (0.53) MAPK8SYK
SCHEMBL7798242 0.66 KDM4E (0.72) MAPK8ALDH1A1KDM4EHPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009140164-A1 6-AMINONICOTINAMIDE DERIVATIVES AS POTENT AND SELECTIVE HISTONE DEACETYLASE INHIBITORS CHIPSCREEN BIOSCIENCES LTD. (CN) 2009-11-19 WO disclosed