SCHEMBL4540972

SCHEMBL4540972

CC(C)(C)OC(=O)N1CCC(C2OCc3cc(-c4ccc(C(=O)N5CCOCC5)cc4)ccc3O2)CC1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 8/20 0.47
ABL1 P00519 1/20 0.46
RIN1 Q13671 1/20 0.46
PTPN2 P17706 1/20 0.44
PTPN1 P18031 1/20 0.44
PTPN6 P29350 1/20 0.44
RECQL P46063 1/20 0.42
CRBN Q96SW2 1/20 0.42
BTK Q06187 1/20 0.41
LMNA P02545 1/20 0.41
USP2 O75604 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HDAC4 P56524 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13586034 0.92 ABL1 (0.46) GPR119ABL1RIN1PTPN2PTPN1
SCHEMBL4347903 0.90 GPR119 (0.44) GPR119RECQLLMNA
SCHEMBL4355169 0.90 PTPN2 (0.44) GPR119ABL1RIN1PTPN2PTPN1
SCHEMBL4536702 0.88 GPR119 (0.49) GPR119PTPN2PTPN1PTPN6
SCHEMBL4521195 0.88 GPR119 (0.42) GPR119PTPN2PTPN1PTPN6RECQL
SCHEMBL4353381 0.88 GPR119 (0.54) GPR119PTPN2PTPN1PTPN6
SCHEMBL4533028 0.86 HPGD (0.41) ABL1RIN1KMT2A
SCHEMBL4360506 0.86 GPR119 (0.47) GPR119PTPN2PTPN1PTPN6
SCHEMBL4353589 0.86 PTPN2 (0.48) GPR119ABL1RIN1PTPN2PTPN1
SCHEMBL4358178 0.85 GPR119 (0.51) GPR119PTPN2PTPN1PTPN6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009150144-A1 NEW GPR119MODULATORS INOVACIA AB (SE) 2009-12-17 WO claimed
WO-2009150144-A1 NEW GPR119MODULATORS INOVACIA AB (SE) 2009-12-17 WO disclosed
WO-2009150144-A1 NEW GPR119MODULATORS INOVACIA AB (SE) 2009-12-17 WO disclosed