SCHEMBL454172

SCHEMBL454172

C=C(Cc1ccc(N)cc1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAOB P27338 8/20 0.48
MAOA P21397 6/20 0.48
CNR2 P34972 1/20 0.40
TSHR P16473 2/20 0.39
CYP3A4 P08684 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
GFER P55789 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LOXL2 Q9Y4K0 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38
HSD17B10 Q99714 1/20 0.38
RAB9A P51151 2/20 0.38
NPC1 O15118 1/20 0.38
GAA P10253 1/20 0.37
MAPT P10636 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
SIGMAR1 Q99720 1/20 0.37
PLAU P00749 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10609924 0.92 MAOB (0.48) MAOBMAOACNR2TSHRCYP3A4
SCHEMBL31503232 0.90 GFER (0.44) MAOBMAOATSHRCYP3A4TDP1
SCHEMBL163962 0.85 MAOA (0.50) MAOBMAOATSHRMAPTL3MBTL1
SCHEMBL11015736 0.82 LMNA (0.55) MAOBMAOATSHRALDH1A1TAAR1
SCHEMBL6546365 0.80 TP53 (0.50) MAOBMAOAALDH1A1RAB9ASMN1; SMN2
SCHEMBL6546799 0.80 L3MBTL1 (0.47) MAOBMAOATDP1RAB9ANPC1
SCHEMBL2448732 0.80 L3MBTL1 (0.52) MAOBMAOATDP1ALDH1A1RAB9A
SCHEMBL6546541 0.79 RAB9A (0.49) MAOBMAOACNR2ALDH1A1RAB9A
SCHEMBL13381339 0.78 TSHR (0.54) TSHRALDH1A1HSD17B10L3MBTL1
SCHEMBL13069103 0.77 SLC6A4 (0.43) MAOBMAOACYP3A4ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 249 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230137331-A1 Activation and Expansion of T Cell Subsets Using Biocompatible Solid Substrates with Tunable Rigidity UNIV PENNSYLVANIA (US) 2023-05-04 US claimed
US-20150030619-A1 Activation and Expansion of T Cell Subsets Using Biocompatible Solid Substrates with Tunable Rigidity THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2015-01-29 US claimed
WO-2013036585-A1 ACTIVATION AND EXPANSION OF T CELL SUBSETS USING BIOCOMPATIBLE SOLID SUBSTRATES WITH TUNABLE RIGIDITY THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2013-03-14 WO claimed
EP-0930844-B8 IMPROVED METHODS FOR DIAGNOSTIC IMAGING BY REGULATING THE ADMINISTRATION RATE OF A CONTRAST AGENT LANTHEUS MEDICAL IMAGING INC (US) 2008-11-26 EP claimed
EP-0930844-B1 IMPROVED METHODS FOR DIAGNOSTIC IMAGING BY REGULATING THE ADMINISTRATION RATE OF A CONTRAST AGENT IMARX PHARMACEUTICAL CORP (US) 2008-09-03 EP claimed
JP-4139440-B2 2008-08-27 JP claimed
EP-0580726-B2 LOW DENSITY MICROSPHERES AND THEIR USE AS CONTRAST AGENTS FOR COMPUTED TOMOGRAPHY IMARX PHARMACEUTICAL CORP (US) 2008-08-20 EP claimed
EP-1017425-B1 IMPROVED METHODS FOR DIAGNOSTIC IMAGING INVOLVING THE USE OF A CONTRAST AGENT AND A CORONARY VASODILATOR IMARX PHARMACEUTICAL CORP (US) 2007-10-17 EP claimed
EP-1323434-B1 Method for diagnostic imaging of the renal region using a contrast agent and a vasodilator IMARX PHARMACEUTICAL CORP (US) 2007-07-11 EP claimed
US-6998107-B2 Composition comprising low density microspheres BRISTOL-MYERS SQUIBB PHARMA COMAPANY (US) 2006-02-14 US claimed
EP-0804932-A2 Contrast media for diagnostic imaging comprising gas filled microspeures ImaRx Pharmaceutical Corp. (US) 1997-11-05 EP claimed
WO-1996040285-A1 NOVEL TARGETED COMPOSITIONS FOR DIAGNOSTIC AND THERAPEUTIC USE IMARX PHARMACEUTICAL CORP. (US) 1996-12-19 WO claimed
US-5547656-A Low density microspheres and their use as contrast agents for computed tomography, and in other applications IMARX PHARMACEUTICAL CORP. (US) 1996-08-20 US claimed
US-5527521-A AQUEOUS SUSPENSION OF BIOCOMPATIBLE POLYMER, A PERFLUOROCARBON GAS, AND A THICKENING OR SUSPENDING AGENT IMARX PHARMACEUTICAL CORP. (US) 1996-06-18 US claimed
US-5456900-A Low density microspheres and their use as contrast agents for computed tomography CITIZENS BANK, N.A. 1995-10-10 US claimed
EP-0580726-A4 LOW DENSITY MICROSPHERES AND THEIR USE AS CONTRAST AGENTS FOR COMPUTED TOMOGRAPHY. UNGER EVAN C (US) 1995-03-29 EP claimed
EP-0580726-A1 LOW DENSITY MICROSPHERES AND THEIR USE AS CONTRAST AGENTS FOR COMPUTED TOMOGRAPHY IMARX PHARMACEUTICAL CORP. (US) 1994-02-02 EP claimed
US-5281408-A Low density microspheres and their use as contrast agents for computed tomography CITIZENS BANK, N.A. 1994-01-25 US claimed
US-5205290-A LOW DENSITY MICROSPHERES AND THEIR USE AS CONTRAST AGENTS FOR COMPUTED TOMOGRAPHY CITIZENS BANK, N.A. 1993-04-27 US claimed
WO-1992017514-A1 LOW DENSITY MICROSPHERES AND THEIR USE AS CONTRAST AGENTS FOR COMPUTED TOMOGRAPHY UNGER EVAN C (US) 1992-10-15 WO claimed