SCHEMBL4542258

SCHEMBL4542258

N[C@@H](Cc1ccc(OC(=O)[C@@H]2CCCN2)cc1)C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.45
SLC7A5 Q01650 4/20 0.44
ITGB3 P05106 1/20 0.44
ITGA2B P08514 1/20 0.44
PTGS1 P23219 3/20 0.43
ALPI P09923 1/20 0.43
PKM P14618 1/20 0.43
XIAP P98170 1/20 0.43
HTR2C P28335 2/20 0.42
HTR2B P41595 1/20 0.42
CTSC P53634 4/20 0.41
CYP3A4 P08684 3/20 0.40
ALOX15 P16050 3/20 0.40
HIF1A Q16665 3/20 0.40
ALDH1A1 P00352 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
TDP1 Q9NUW8 2/20 0.40
KDM4E B2RXH2 2/20 0.40
ABCB11 O95342 1/20 0.40
CHRM2 P08172 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Proline SCHEMBL17728310 0.96 PTPN1 (0.43) PTPN1SLC7A5ITGB3ITGA2BPTGS1
Threonine SCHEMBL17728293 0.89 SLC7A5 (0.37) PTPN1SLC7A5ITGB3ITGA2BPTGS1
Proline SCHEMBL17728296 0.88 HTR2C (0.37) PTPN1SLC7A5ITGB3ITGA2BPTGS1
SCHEMBL3100802 0.88 ITGB3 (0.38) PTPN1SLC7A5ITGB3ITGA2BPTGS1
Alanine SCHEMBL1826638 0.88 SLC7A5 (0.37) PTPN1SLC7A5ITGB3ITGA2BPTGS1
SCHEMBL17728295 0.88 HTR2C (0.36) PTPN1SLC7A5ITGB3ITGA2BPTGS1
SCHEMBL5576438 0.87 SLC7A5 (0.41) PTPN1SLC7A5ITGB3ITGA2BPTGS1
SCHEMBL1675509 0.86 SLC7A5 (0.44) PTPN1SLC7A5ITGB3ITGA2BHTR2C
Tyrosine SCHEMBL4352798 0.84 SLC7A5 (0.57) PTPN1SLC7A5PTGS1ALPIPKM
SCHEMBL6284117 0.83 SLC7A5 (0.46) PTPN1SLC7A5ITGB3ITGA2BPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112813064-A Method for creating endogenous herbicide-resistant rice with high and stable resistance 安徽省农业科学院水稻研究所 2021-05-18 CN disclosed
WO-2020245748-A1 METHODS AND SYSTEMS FOR ASSESSING A PHENOTYPE OF A BIOLOGICAL TISSUE OF A PATIENT USING RAMAN SPECTROSCOPY POLYVALOR, LIMITED PARTNERSHIP (CA) 2020-12-10 WO disclosed
WO-2012062906-A1 PEPTIDES AS BIOACTIVE COMPOUNDS INSTITUTO BIOMAR, S.A. (ES) 2012-05-18 WO disclosed
EP-1202963-B1 SPLA2 INHIBITORS LILLY CO ELI (US) 2007-01-03 EP disclosed
US-6900238-B1 HIV protease inhibitors THE SCRIPPS RESEARCH INSTITUTE (US) 2005-05-31 US disclosed
EP-0873519-A4 HIV PROTEASE INHIBITORS SCRIPPS RESEARCH INST (US) 2005-04-27 EP disclosed
EP-0873519-A1 HIV PROTEASE INHIBITORS The Scripps Research Institute (US) 1998-10-28 EP disclosed
WO-1997021100-A9 HIV PROTEASE INHIBITORS 1997-10-30 WO disclosed
WO-1997021100-A1 HIV PROTEASE INHIBITORS THE SCRIPPS RESEARCH INSTITUTE (US) 1997-06-12 WO disclosed
US-4473646-A SEPARATION OF ISOMERS, PURIFICATION DEVELOPMENT FINANCE CORP. OF NEW ZEALAND (NZ) 1984-09-25 US disclosed
US-4064235-A INCREASING RENAL BLOOD FLOW EISAI CO., LTD. (JA) 1977-12-20 US disclosed
US-4064235-A INCREASING RENAL BLOOD FLOW EISAI CO., LTD. (JA) 1977-12-20 US disclosed