SCHEMBL6284117

SCHEMBL6284117

NC(=O)[C@@H]1CCCN1.N[C@@H](Cc1ccc(OC(=O)[C@@H](N)Cc2ccccc2)cc1)C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC7A5 Q01650 3/20 0.46
ALPI P09923 1/20 0.46
PKM P14618 1/20 0.46
PTGS1 P23219 1/20 0.46
XIAP P98170 1/20 0.46
HTR2C P28335 1/20 0.44
HTR2B P41595 1/20 0.44
CTSC P53634 2/20 0.43
DPP4 P27487 5/20 0.40
DPP8 Q6V1X1 4/20 0.40
DPP9 Q86TI2 4/20 0.40
DPP7 Q9UHL4 4/20 0.40
PTPN1 P18031 1/20 0.40
TACR1 P25103 1/20 0.39
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
FAP Q12884 3/20 0.38
KCNH2 Q12809 1/20 0.38
TPH1 P17752 1/20 0.38
TYR P14679 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10757105 0.86 HTR2C (0.45) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL29131638 0.86 CTSC (0.46) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL4542258 0.83 PTPN1 (0.45) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL5576438 0.82 SLC7A5 (0.41) SLC7A5ALPIPKMPTGS1XIAP
Proline SCHEMBL28237451 0.82 PTPN1 (0.38) SLC7A5ALPIPKMPTGS1XIAP
SCHEMBL1003560 0.82 SLC7A5 (0.69) SLC7A5ALPIPKMPTGS1XIAP
Phenylalanine SCHEMBL5699042 0.82 SLC7A5 (0.69) SLC7A5ALPIPKMPTGS1XIAP
Phenylalanine SCHEMBL5608077 0.82 SLC7A5 (0.69) SLC7A5ALPIPKMPTGS1XIAP
D-Phenylalanine SCHEMBL2184336 0.81 SLC7A5 (0.59) SLC7A5ALPIPKMPTGS1XIAP
Dl-Phenylalanine SCHEMBL498385 0.81 SLC7A5 (0.59) SLC7A5ALPIPKMPTGS1XIAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6900238-B1 HIV protease inhibitors THE SCRIPPS RESEARCH INSTITUTE (US) 2005-05-31 US disclosed
EP-0873519-A4 HIV PROTEASE INHIBITORS SCRIPPS RESEARCH INST (US) 2005-04-27 EP disclosed
EP-0873519-A1 HIV PROTEASE INHIBITORS The Scripps Research Institute (US) 1998-10-28 EP disclosed
WO-1997021100-A9 HIV PROTEASE INHIBITORS 1997-10-30 WO disclosed
WO-1997021100-A1 HIV PROTEASE INHIBITORS THE SCRIPPS RESEARCH INSTITUTE (US) 1997-06-12 WO disclosed