SCHEMBL4542554

SCHEMBL4542554

O=C(NCCC1CCN(S(=O)(=O)c2ccc(Cl)cc2)C1)C12CC3CC(CC(C3)C1)C2

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.51
DRD4 P21917 2/20 0.51
LMNA P02545 1/20 0.49
TSHR P16473 1/20 0.49
ALOX12 P18054 1/20 0.49
HTT P42858 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
ALDH1A1 P00352 4/20 0.45
POLB P06746 1/20 0.45
GAA P10253 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
EPHX2 P34913 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4534658 0.90 CYP3A4 (0.49) ALDH1A1POLBMEN1KMT2A
SCHEMBL4539521 0.90 ALDH1A1 (0.46) LMNATSHRNPSR1ALDH1A1POLB
SCHEMBL8061563 0.90 LMNA (0.51) DRD2DRD4LMNATSHRALOX12
SCHEMBL4538134 0.90 ALDH1A1 (0.48) LMNAALDH1A1GAAMEN1KMT2A
SCHEMBL4535269 0.90 LMNA (0.51) DRD2DRD4LMNATSHRALOX12
SCHEMBL4542877 0.88 HSD11B1 (0.44) DRD2DRD4ALDH1A1MEN1KMT2A
SCHEMBL4541776 0.85 LMNA (0.55) DRD2DRD4LMNATSHRALOX12
SCHEMBL4541025 0.85 MEN1 (0.50) DRD2DRD4LMNATSHRALOX12
SCHEMBL4541325 0.84 HDAC3 (0.50) DRD2DRD4EPHX2
SCHEMBL4541251 0.82 EPHX2 (0.45) LMNAALDH1A1POLBGAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO claimed
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed