SCHEMBL4542802

SCHEMBL4542802

COCCN/C(=N\C#N)N1CCC(CC(N)C(=O)N(O)S(=O)(=O)c2cc(F)c(Oc3ccc(F)cc3)c(F)c2)CC1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.33
SLC9A3 P48764 3/20 0.33
RORC P51449 2/20 0.32
HTR2A P28223 2/20 0.31
KMT2A Q03164 2/20 0.30
MEN1 O00255 1/20 0.30
MMP1 P03956 1/20 0.30
MMP13 P45452 1/20 0.30
ALDH1A1 P00352 1/20 0.30
RAB9A P51151 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4374211 0.89 SLC9A3 (0.35) NPC1SLC9A3RORCHTR2AKMT2A
SCHEMBL1799220 0.82 ADAMTS7 (0.45) NPC1SLC9A3RORCMMP1MMP13
SCHEMBL1799218 0.82 ADAMTS7 (0.45) NPC1SLC9A3RORCMMP1MMP13
SCHEMBL4372629 0.78 PKM (0.41) KMT2AMEN1MMP1MMP13ALDH1A1
SCHEMBL4288103 0.75 MMP3 (0.41) KMT2AMEN1MMP1MMP13ALDH1A1
SCHEMBL4288106 0.75 MMP3 (0.41) KMT2AMEN1MMP1MMP13ALDH1A1
SCHEMBL3875819 0.74 SLC9A3 (0.41) NPC1SLC9A3ALDH1A1RAB9A
SCHEMBL4376127 0.72 L3MBTL1 (0.39) MMP1MMP13
SCHEMBL1800636 0.69 ADAMTS7 (0.48) MMP1MMP13
SCHEMBL1800637 0.69 ADAMTS7 (0.48) MMP1MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1461313-B1 HUMAN ADAM-10 INHIBITORS EXELIXIS INC (US) 2009-08-05 EP disclosed