SCHEMBL4543095

SCHEMBL4543095

CC(C)(C(=O)O)c1ccc(N2CCN(c3ccc(-c4nc5cc(Cl)ccc5[nH]4)cn3)CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 17/20 0.53
KCNH2 Q12809 11/20 0.53
ADORA2A P29274 3/20 0.51
SOAT1 P35610 3/20 0.46
CHEK2 O96017 2/20 0.45
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4559775 0.91 DGAT1 (0.49) DGAT1KCNH2ADORA2ASOAT1CHEK2
SCHEMBL6994712 0.84 DGAT1 (0.54) DGAT1KCNH2ADORA2ACHEK2CYP2C9
SCHEMBL4561989 0.84 DGAT1 (0.56) DGAT1KCNH2ADORA2ACHEK2CYP3A4
SCHEMBL6995932 0.84 DGAT1 (0.51) DGAT1KCNH2ADORA2ASOAT1CYP2C9
SCHEMBL4543375 0.84 CHEK2 (0.59) DGAT1KCNH2ADORA2ACHEK2CYP2C9
SCHEMBL4562539 0.82 DGAT1 (0.54) DGAT1KCNH2ADORA2ACHEK2CYP3A4
SCHEMBL6993769 0.82 CHEK2 (0.53) DGAT1KCNH2ADORA2ACHEK2CYP2C9
SCHEMBL4538780 0.81 DGAT1 (0.51) DGAT1KCNH2ADORA2ACHEK2CYP2C9
SCHEMBL4560992 0.81 DGAT1 (0.57) DGAT1KCNH2ADORA2ASOAT1CHEK2
SCHEMBL10081917 0.81 DGAT1 (0.51) DGAT1KCNH2ADORA2ASOAT1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064569-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-05-18 WO disclosed
WO-2012064569-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-05-18 WO disclosed