SCHEMBL4543375

SCHEMBL4543375

NC(=O)c1ccc(N2CCN(c3ccc(-c4nc5cc(Cl)ccc5[nH]4)cn3)CC2)cc1

nearest known ligand 0.59

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 9/20 0.59
DGAT1 O75907 9/20 0.54
KCNH2 Q12809 6/20 0.54
ADORA2A P29274 2/20 0.54
MGLL Q99685 1/20 0.47
CYP2C9 P11712 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4560928 0.93 DGAT1 (0.54) CHEK2DGAT1KCNH2ADORA2AMGLL
SCHEMBL4538780 0.88 DGAT1 (0.51) CHEK2DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL4560992 0.86 DGAT1 (0.57) CHEK2DGAT1KCNH2ADORA2AMGLL
SCHEMBL4561989 0.85 DGAT1 (0.56) CHEK2DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL6994712 0.85 DGAT1 (0.54) CHEK2DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL4543095 0.84 DGAT1 (0.53) CHEK2DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL4562539 0.84 DGAT1 (0.54) CHEK2DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL6993769 0.83 CHEK2 (0.53) CHEK2DGAT1KCNH2ADORA2AMGLL
SCHEMBL4562113 0.83 DGAT1 (0.52) DGAT1KCNH2ADORA2ACYP2C9
SCHEMBL4559775 0.82 DGAT1 (0.49) CHEK2DGAT1KCNH2ADORA2ACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012064569-A1 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-05-18 WO disclosed