Fludrocortisone

Fludrocortisone

SCHEMBL4545

C[C@]12CCC(=O)C=C1CC[C@H]1[C@@H]3CC[C@](O)(C(=O)CO)[C@@]3(C)C[C@H](O)[C@@]12F

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 7/20 1.00
PGR P06401 4/20 0.78
HIF1A Q16665 4/20 0.78
HRH1 P35367 1/20 0.78
SERPINA6 P08185 3/20 0.76
HSD17B10 Q99714 4/20 0.73
AR P10275 3/20 0.73
ALDH1A1 P00352 1/20 0.68
MAPK1 P28482 1/20 0.68
FNTA P49354 1/20 0.68
FNTB P49356 1/20 0.68
LMNA P02545 2/20 0.64
CYP2C19 P33261 3/20 0.61
CYP3A4 P08684 4/20 0.58
SHBG P04278 2/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
NR3C2 P08235 1/20 0.58
MAPT P10636 1/20 0.58
NFKB1 P19838 1/20 0.58
KMT2A Q03164 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fludrocortisone SCHEMBL10598529 1.00 NR3C1 (1.00) NR3C1PGRHIF1AHRH1SERPINA6
Fludrocortisone SCHEMBL19327146 1.00 NR3C1 (1.00) NR3C1PGRHIF1AHRH1SERPINA6
Fludrocortisone SCHEMBL5188889 1.00 NR3C1 (1.00) NR3C1PGRHIF1AHRH1SERPINA6
Fludrocortisone SCHEMBL14373312 1.00 NR3C1 (1.00) NR3C1PGRHIF1AHRH1SERPINA6
Fludrocortisone SCHEMBL4323075 1.00 NR3C1 (1.00) NR3C1PGRHIF1AHRH1SERPINA6
Fludrocortisone SCHEMBL13026141 1.00 NR3C1 (1.00) NR3C1PGRHIF1AHRH1SERPINA6
Fludrocortisone SCHEMBL23975175 1.00 NR3C1 (1.00) NR3C1PGRHIF1AHRH1SERPINA6
Fludrocortisone SCHEMBL21297043 0.98 NR3C1 (0.96) NR3C1PGRHIF1AHRH1SERPINA6
SCHEMBL8735123 0.93 NR3C1 (0.87) NR3C1PGRHIF1AHRH1SERPINA6
SCHEMBL8735124 0.93 NR3C1 (0.87) NR3C1PGRHIF1AHRH1SERPINA6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 24912 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4747263-A1 LIPID NANOPARTICLES AND USES THEREOF University of Connecticut (US) 2026-05-27 EP claimed
CN-116209439-B Cereblon protein modulators Saint Jude Children's Research Hospital Ltd. (US) 2026-05-26 CN claimed
WO-2026102485-A1 PRODUCTS AND METHODS FOR THE ASSESSMENT AND TREATMENT OF SEPSIS AND IMMUNOLOGICAL AND INFLAMMATORY CONDITIONS CENTRAL ADELAIDE LOCAL HEALTH NETWORK INC (AU) 2026-05-21 WO claimed
US-20260139030-A1 CHIMERIC PROTEINS FOR TREATING CUTANEOUS INFLAMMATION SHATTUCK LABS INC (US) 2026-05-21 US claimed
WO-2026100654-A1 NUCLEIC ACID INTRODUCTION AID, NUCLEIC ACID INTRODUCTION AGENT, AND NUCLEIC ACID INTRODUCTION METHOD 株式会社インファーマシア 2026-05-15 WO claimed
US-20260125650-A1 METHODS AND COMPOSITIONS FOR GENERATING HEPATOCYTES TRAILHEAD BIOSYSTEMS INC (US) 2026-05-07 US claimed
WO-2026087695-A1 TREATMENT FOR METABOLIC DISORDER SAPREME TECHNOLOGIES B.V. (NL) 2026-04-30 WO claimed
US-20260108610-A1 Drug-Resistant Immune Cells and Methods of Use Thereof REGENTS OF THE UNIVERSITY OF MINNESOTA 2026-04-23 US claimed
US-20260109699-A1 AZOLE DERIVATIVES AS SHP2 INHIBITORS IRBM S.P.A. (IT) 2026-04-23 US claimed
EP-4728280-A1 COMPOUNDS FOR DIAGNOSING AND TREATING EPILEPSY SYNDROMES, METHODS AND USES THEREOF BIOSTRIKE UNIPESSOAL LDA (PT) 2026-04-22 EP claimed
EP-0055870-A1 Pyridylmethyl esters of selected bio-affecting carboxylic acids, process for preparing and pharmaceutical composition comprising the same MERCK & CO. INC. (US) 1982-07-14 EP claimed
EP-0051278-A1 Soft tertiary amine esters of bio-affecting carboxylic acids, processes for preparing and a pharmaceutical composition containing the same MERCK & CO. INC. (US) 1982-05-12 EP claimed
EP-0033341-A1 CYTOTOXIC NUCLEOSIDE-CORTICOSTEROID PHOSPHODIESTERS Research Corporation (US) 1981-08-12 EP claimed
US-4283394-A ANTICARCINOGENIC AGENTS RESEARCH CORPORATION (US) 1981-08-11 US claimed
US-4279900-A ANTIINFLAMMATORY INTREX RESEARCH CORPORATION (US) 1981-07-21 US claimed
EP-0028110-A2 Autoclavable emulsions Smith and Nephew Associated Companies p.l.c. (GB) 1981-05-06 EP claimed
WO-1981000410-A1 CYTOTOXIC NUCLEOSIDE-CORTICOSTEROID PHOSPHODIESTERS RESEARCH CORP (US) 1981-02-19 WO claimed
US-4137311-A CORTICOSTEROIDS, METAL ADDUCTS OF BIS(2-PYRIDYL-1-OXIDE)-DISULFIDE; DERMATITIS, ANTIINFLAMMATORY WILLIAM H. RORER, INC. (US) 1979-01-30 US claimed
US-4083974-A Topical steroidal anti-inflammatory preparations containing polyoxypropylene 15 stearyl ether THE UPJOHN COMPANY (US) 1978-04-11 US claimed
US-4041055-A SULFENYLATION, MICHAEL ADDITION, REACTION WITH THIOPHILE, HYDROLYSIS THE UPJOHN COMPANY (US) 1977-08-09 US claimed