SCHEMBL4547659

SCHEMBL4547659

Cc1c(F)cc(CBr)cc1F

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
TRPA1 O75762 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22817324 0.86 CYP1A2 (0.33) HDAC1HDAC6
SCHEMBL15241715 0.78 RAPGEF4 (0.35)
SCHEMBL28880200 0.78 HMGB1 (0.40) HDAC1HDAC6ALDH1A1
SCHEMBL13932538 0.78 HDAC1 (0.38) HDAC1HDAC6
SCHEMBL391029 0.78 CES2 (0.36) TRPA1ALDH1A1TSHR
SCHEMBL18553018 0.78 PTGS1 (0.40) HDAC1HDAC6
SCHEMBL24357406 0.77
SCHEMBL30626589 0.77
SCHEMBL24357673 0.76 KDM1A (0.37) TRPA1ALDH1A1TSHR
SCHEMBL6886890 0.76 HDAC1 (0.37) HDAC1HDAC6TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250243205-A1 sGC STIMULATORS TISENTO THERAPEUTICS INC (US) 2025-07-31 US disclosed
US-20250059197-A1 sGC STIMULATORS TISENTO THERAPEUTICS INC (US) 2025-02-20 US disclosed
US-11897887-B2 sGC stimulators TISENTO THERAPEUTICS INC. (US) 2024-02-13 US disclosed
CN-111712247-B sGC stimulators 塞科里昂医疗股份有限公司 2024-02-09 CN disclosed
EP-3342766-B1 SMALL MOLECULE COMPOUND FOR ENHANCING PLANT STRESS RESISTANCE CAS CENTER FOR EXCELLENCE IN MOLECULAR PLANT SCIENCES (CN) 2020-12-09 EP disclosed
US-20200377508-A1 sGC STIMULATORS TISENTO THERAPEUTICS INC. 2020-12-03 US disclosed
US-10842151-B2 Small molecule compound for enhancing plant stress resistance CAS CENTER FOR EXCELLENCE IN MOLECULAR PLANT SCIENCES (CN) 2020-11-24 US disclosed
EP-3727388-A1 SGC STIMULATORS Cyclerion Therapeutics, Inc. (US) 2020-10-28 EP disclosed
CN-111712247-A sGC stimulators 塞科里昂医疗股份有限公司 2020-09-25 CN disclosed
US-20180360039-A1 Small Molecule Compound for Enhancing Plant Stress Resistance CAS CENTER FOR EXCELLENCE IN MOLECULAR PLANT SCIENCES (CN) 2018-12-20 US disclosed
EP-3342766-A1 SMALL MOLECULE COMPOUND FOR ENHANCING PLANT STRESS RESISTANCE Shanghai Institutes for Biological Sciences, Chinese Academy of Sciences (CN) 2018-07-04 EP disclosed
US-8173704-B2 Difluorophenol derivatives and their use BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2012-05-08 US disclosed
US-20090291993-A1 Difluorophenol Derivatives and Their Use BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2009-11-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250059197-A1 sGC STIMULATORS GMPS, GUCY1A2, PDE2A HDAC1 3330/4885HDAC6 3716/4885TRPA1 2486/4885
US-20090291993-A1 Difluorophenol Derivatives and Their Use TPMT, FABP3, DPP4 HDAC1 1744/4885HDAC6 1012/4885TRPA1 3762/4885
US-11897887-B2 sGC stimulators GMPS, GUCY1A2, PDE2A HDAC1 3404/4885HDAC6 3836/4885TRPA1 2400/4885
US-10842151-B2 Small molecule compound for enhancing plant stress resistance CYP4F11, RICTOR, MYB HDAC1 1165/4885HDAC6 2131/4885TRPA1 256/4885
US-20200377508-A1 sGC STIMULATORS GMPS, GUCY1A2, PDE2A HDAC1 3404/4885HDAC6 3836/4885TRPA1 2400/4885
US-20180360039-A1 Small Molecule Compound for Enhancing Plant Stress Resistance CYP4F11, RICTOR, MYB HDAC1 1165/4885HDAC6 2131/4885TRPA1 256/4885
US-20250243205-A1 sGC STIMULATORS GMPS, GUCY1A2, PDE2A HDAC1 3330/4885HDAC6 3716/4885TRPA1 2486/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.