SCHEMBL454901

SCHEMBL454901

Clc1[c]c(Br)c(-c2ccccc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.41
MAPK1 P28482 3/20 0.41
CYP2A6 P11509 1/20 0.41
CTRC Q99895 2/20 0.37
CSNK2A1 P68400 2/20 0.35
CYP1A2 P05177 1/20 0.34
BACE1 P56817 1/20 0.33
ALOX5 P09917 1/20 0.33
HSD17B10 Q99714 2/20 0.32
HPGD P15428 1/20 0.32
BCL2L1 Q07817 1/20 0.32
PTGS2 P35354 1/20 0.31
ESR2 Q92731 1/20 0.31
AKR1C3 P42330 1/20 0.30
AKR1C2 P52895 1/20 0.30
AKR1C1 Q04828 1/20 0.30
TP53 P04637 1/20 0.30
MAPT P10636 1/20 0.30
NFKB1 P19838 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL456350 0.78 CYP2A6 (0.44) ALDH1A1MAPK1CYP2A6CTRCCSNK2A1
SCHEMBL457364 0.78 ALDH1A1 (0.44) ALDH1A1MAPK1CYP2A6CTRCBACE1
SCHEMBL457904 0.75 CYP2A6 (0.41) ALDH1A1MAPK1CYP2A6CTRCCSNK2A1
SCHEMBL457524 0.75 ALDH1A1 (0.41) ALDH1A1MAPK1CYP2A6BACE1ALOX5
SCHEMBL7814278 0.75 CYP2A6 (0.41) ALDH1A1MAPK1CYP2A6CTRCCSNK2A1
SCHEMBL6206554 0.75 CYP2A6 (0.41) ALDH1A1CYP2A6CTRCCSNK2A1CYP1A2
SCHEMBL455577 0.71 ALDH1A1 (0.41) ALDH1A1MAPK1CYP2A6CTRCCSNK2A1
SCHEMBL21053453 0.71 CSNK2A1 (0.47) ALDH1A1MAPK1CYP2A6CTRCCSNK2A1
SCHEMBL456752 0.71 CYP2A6 (0.38) CYP2A6CTRCCSNK2A1CYP1A2BACE1
SCHEMBL457102 0.71 ALDH1A1 (0.38) ALDH1A1MAPK1BACE1ALOX5ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614053-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2013-07-17 EP disclosed
WO-2012033225-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-03-15 WO disclosed