SCHEMBL457364

SCHEMBL457364

Brc1[c]c(Br)c(-c2ccccc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.44
MAPK1 P28482 4/20 0.44
BACE1 P56817 1/20 0.36
ALOX5 P09917 1/20 0.35
HSD17B10 Q99714 2/20 0.34
HPGD P15428 1/20 0.34
BCL2L1 Q07817 1/20 0.34
CYP2A6 P11509 1/20 0.34
ESR2 Q92731 1/20 0.32
TDO2 P48775 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32
AKR1C1 Q04828 1/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
NFKB1 P19838 1/20 0.32
RAB9A P51151 1/20 0.32
NFKB2 Q00653 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL457524 0.78 ALDH1A1 (0.41) ALDH1A1MAPK1BACE1ALOX5HSD17B10
SCHEMBL455577 0.78 ALDH1A1 (0.41) ALDH1A1MAPK1BACE1ALOX5HSD17B10
SCHEMBL454901 0.78 ALDH1A1 (0.41) ALDH1A1MAPK1BACE1ALOX5HSD17B10
SCHEMBL456919 0.78 ALDH1A1 (0.41) ALDH1A1MAPK1BACE1ALOX5HSD17B10
SCHEMBL456995 0.78 ALDH1A1 (0.41) ALDH1A1MAPK1BACE1ALOX5HSD17B10
SCHEMBL7736209 0.78
SCHEMBL455612 0.74 ALDH1A1 (0.38) ALDH1A1MAPK1BACE1L3MBTL1TP53
SCHEMBL457102 0.74 ALDH1A1 (0.38) ALDH1A1MAPK1BACE1ALOX5ESR2
SCHEMBL459103 0.72 ALDH1A1 (0.36) ALDH1A1MAPK1HSD17B10HPGDMAPT
SCHEMBL25862086 0.69 ALDH1A1 (0.57) ALDH1A1MAPK1BACE1ALOX5HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614053-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2013-07-17 EP disclosed
WO-2012033225-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-03-15 WO disclosed