SCHEMBL457524

SCHEMBL457524

Cc1[c]c(Br)c(-c2ccccc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.41
MAPK1 P28482 2/20 0.41
ESR2 Q92731 1/20 0.38
CYP2A6 P11509 2/20 0.36
CYP2B6 P20813 1/20 0.36
AKT1 P31749 1/20 0.34
AKT2 P31751 1/20 0.34
BACE1 P56817 1/20 0.33
ALOX5 P09917 1/20 0.33
PDCD1 Q15116 1/20 0.33
CD274 Q9NZQ7 1/20 0.33
AURKA O14965 1/20 0.32
AURKB Q96GD4 1/20 0.32
HSD17B10 Q99714 2/20 0.32
HPGD P15428 2/20 0.32
BCL2L1 Q07817 1/20 0.32
MAOB P27338 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
PSMB5 P28074 1/20 0.32
TDO2 P48775 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL457364 0.78 ALDH1A1 (0.44) ALDH1A1MAPK1ESR2CYP2A6BACE1
SCHEMBL4371389 0.78 ESR2 (0.41) ALDH1A1MAPK1ESR2CYP2A6CYP2B6
SCHEMBL454901 0.75 ALDH1A1 (0.41) ALDH1A1MAPK1ESR2CYP2A6BACE1
SCHEMBL12503755 0.75 CYP2A6 (0.41) ALDH1A1ESR2CYP2A6CYP2B6AKT1
SCHEMBL14675940 0.75 ESR2 (0.38) ALDH1A1MAPK1ESR2CYP2A6CYP2B6
SCHEMBL457819 0.75 ESR2 (0.38) ALDH1A1MAPK1ESR2CYP2A6CYP2B6
SCHEMBL457102 0.75 ALDH1A1 (0.38) ALDH1A1MAPK1ESR2BACE1ALOX5
SCHEMBL456629 0.72 SQOR (0.39) ALDH1A1ESR2CYP2A6CYP2B6BACE1
SCHEMBL456995 0.71 ALDH1A1 (0.41) ALDH1A1MAPK1ESR2CYP2A6CYP2B6
SCHEMBL459103 0.69 ALDH1A1 (0.36) ALDH1A1MAPK1HSD17B10HPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614053-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY LIMITED (JP) 2013-07-17 EP disclosed
WO-2012033225-A1 METHOD FOR PRODUCING PYRIDAZINONE COMPOUNDS AND INTERMEDIATE THEREOF SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2012-03-15 WO disclosed