SCHEMBL4553231

SCHEMBL4553231

NC(=O)c1nc(-c2ccccc2)cn1C(F)(F)F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.48
MAPT P10636 3/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
KDM4E B2RXH2 7/20 0.42
ALDH1A1 P00352 6/20 0.42
HPGD P15428 3/20 0.42
HSD17B10 Q99714 2/20 0.42
MAPK1 P28482 1/20 0.42
MAP2K3 P46734 1/20 0.42
CASP1 P29466 2/20 0.40
TSHR P16473 2/20 0.40
GAA P10253 1/20 0.40
CASP7 P55210 1/20 0.40
PARP1 P09874 2/20 0.39
PKM P14618 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
LIMK1 P53667 1/20 0.39
LMNA P02545 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12907953 0.76 SCN9A (0.61) SCN9AMAPTNPC1RAB9AKDM4E
SCHEMBL9980597 0.71 ALDH1A1 (0.53) MAPTNPC1RAB9AKDM4EALDH1A1
SCHEMBL11890089 0.66 NPC1 (0.49) MAPTNPC1RAB9AKDM4EALDH1A1
SCHEMBL6861398 0.66 TLR8 (0.50) MAPTNPC1RAB9AKDM4EALDH1A1
SCHEMBL28235655 0.65 PARP1 (0.53) MAPTNPC1RAB9AKDM4EALDH1A1
Lithium SCHEMBL31133404 0.65 SCN9A (0.46) SCN9AMAPTNPC1RAB9AKDM4E
SCHEMBL7444775 0.64 SCN9A (0.63) SCN9AMAPTKDM4EMAPK1PARP1
SCHEMBL31460615 0.64 ALDH1A1 (0.60) MAPTNPC1RAB9AKDM4EALDH1A1
Trifluoroacetic Acid SCHEMBL16699728 0.64 ALDH1A1 (0.44) SCN9AMAPTNPC1RAB9AKDM4E
SCHEMBL4553234 0.64 PTGS2 (0.48) MAPK1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009072643-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-06-11 WO disclosed