SCHEMBL4553418

SCHEMBL4553418

Cc1cccc(C(I)(NC(=O)OC(C)(C)C)C2CCC(=O)C2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 1/20 0.39
CCKBR P32239 1/20 0.34
RXFP1 Q9HBX9 1/20 0.33
POLB P06746 1/20 0.33
HSD11B1 P28845 1/20 0.33
KDM1A O60341 1/20 0.33
MAOB P27338 1/20 0.33
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
LMNA P02545 2/20 0.32
NPY2R P49146 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
RORC P51449 1/20 0.32
MAPT P10636 1/20 0.32
ATM Q13315 1/20 0.32
NFKB1 P19838 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17018582 0.74 CYP2C19 (0.44) GPR119RXFP1POLBLMNAMEN1
SCHEMBL4597509 0.73 LMNA (0.40) RXFP1POLBLMNANPSR1MEN1
SCHEMBL1558558 0.72 KCNA3 (0.39) GPR119KDM1AMAOBMEN1KMT2A
SCHEMBL4437715 0.71 GPR119 (0.36) GPR119CCKBRLMNANPSR1MEN1
SCHEMBL1557162 0.68 NFKB1 (0.40) KDM1AMAOBKMT2ANFKB1NFKB2
SCHEMBL3726743 0.64 GAA (0.42) RXFP1POLBLMNAMEN1KMT2A
SCHEMBL5394420 0.64 KDM1A (0.42) GPR119KDM1AMAOBMEN1KMT2A
SCHEMBL17330297 0.63 CHRM3 (0.42) KMT2AMAPT
SCHEMBL8966117 0.63 HSD17B10 (0.59) RXFP1NPSR1MEN1KMT2AMAPT
SCHEMBL29991501 0.63 HSD17B10 (0.59) RXFP1NPSR1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2124913-A1 1-AMINOMETHYL- L- PHENYL- CYCLOHEXANE DERIVATIVES AS DDP-IV INHIBITORS Novartis AG (CH) 2009-12-02 EP disclosed
WO-2008077597-A1 1-AMINOMETHYL- L- PHENYL- CYCLOHEXANE DERIVATIVES AS DDP-IV INHIBITORS NOVARTIS AG (CH) 2008-07-03 WO disclosed